SCHEMBL6538947

SCHEMBL6538947

COC(=O)C[C@H](NC(=O)OCc1ccccc1)NC(=O)[C@@H]1CC=CCN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.44
BACE1 P56817 1/20 0.42
SYK P43405 1/20 0.41
YAP1 P46937 1/20 0.41
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
P2RX7 Q99572 6/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CTSL P07711 1/20 0.39
STS P08842 1/20 0.39
MAPK1 P28482 1/20 0.39
ABCB1 P08183 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CASP1 P29466 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6540111 0.85 ITGB3 (0.52) HTTBACE1SYKYAP1ITGB3
SCHEMBL6538950 0.81 NPC1 (0.43) HTTBACE1SYKYAP1ITGB3
SCHEMBL6939589 0.80 ITGB3 (0.57) HTTYAP1ITGB3ITGA2B
SCHEMBL6539427 0.80 ITGB3 (0.57) HTTYAP1ITGB3ITGA2B
SCHEMBL6935798 0.80 ITGB3 (0.57) HTTYAP1ITGB3ITGA2B
SCHEMBL6539630 0.80 ITGB3 (0.57) HTTYAP1ITGB3ITGA2B
SCHEMBL6936346 0.75 ITGB3 (0.57) YAP1ITGB3ITGA2B
SCHEMBL6943036 0.74 ITGB3 (0.49) HTTYAP1ITGB3ITGA2BNPC1
SCHEMBL8297504 0.74 HTT (0.61) HTTBACE1SYKYAP1ITGB3
SCHEMBL15898105 0.74 SYK (0.49) HTTBACE1SYKYAP1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6812235-B2 2-ACYLAMINO- BETA -ALANINE DERIVATIVES AND A PHARMACEUTICALLY ACCEPTABLE SALT, USEFUL AS FIBRINOGEN RECEPTOR ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-11-02 US disclosed
US-20030018193-A1 Beta-alanine derivatives and their use as receptor anatgonists ASTELLAS PHARMA INC. (JP) 2003-01-23 US disclosed
EP-1255748-A1 BETA-ALANINE DERIVATIVES AND THEIR USE AS RECEPTOR ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-11-13 EP disclosed
WO-2001060813-A1 BETA-ALANINE DERIVATIVES AND THEIR USE AS RECEPTOR ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-08-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030018193-A1 Beta-alanine derivatives and their use as receptor anatgonists ARRB1, ADRB1, GLRB HTT 3050/4885BACE1 540/4885SYK 2740/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.