SCHEMBL6539718

SCHEMBL6539718

COC(=O)Nc1ccc(NC(=O)Nc2ccc(C[C@@H](CO)NC[C@@H](COc3ccccc3)OC(=O)C(F)(F)F)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 15/20 0.61
ADRB1 P08588 13/20 0.61
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
HPGD P15428 1/20 0.37
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6539734 0.96 ADRB3 (0.62) ADRB3ADRB1SMN1; SMN2NPC1RAB9A
SCHEMBL6539720 0.95 ADRB3 (0.60) ADRB3ADRB1SMN1; SMN2NPC1RAB9A
SCHEMBL7532289 0.89 ADRB3 (0.58) ADRB3ADRB1
SCHEMBL6541344 0.89 ADRB3 (0.58) ADRB3ADRB1NPC1RAB9A
SCHEMBL6539506 0.89 ADRB3 (0.59) ADRB3ADRB1NPC1RAB9A
SCHEMBL6539488 0.88 ADRB3 (0.57) ADRB3ADRB1SMN1; SMN2NPC1RAB9A
SCHEMBL6539964 0.88 ADRB3 (0.57) ADRB3ADRB1
Trifluoroacetic Acid SCHEMBL6538892 0.87 ADRB3 (0.79) ADRB3ADRB1
SCHEMBL7533764 0.87 ADRB3 (0.58) ADRB3ADRB1
SCHEMBL6538790 0.86 ADRB3 (0.56) ADRB3ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6826033-B2 BETA 3 ADRENERGIC RECEPTOR AGONISTS; TREATMENT OF POLLAKIURIA, URINARY INCONTINENCE, OBESITY OR DIABETES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-11-30 US disclosed
WO-2002024635-A2 AMINOALCOHOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-03-28 WO disclosed