SCHEMBL6540029

SCHEMBL6540029

CC(C)(C)OC(=O)N(C[C@@H](O)c1cccc(Cl)c1)[C@H](CO)Cc1ccc(NC(=O)c2c[nH]cc2-c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.53
ADRB3 P13945 10/20 0.42
ITGB1 P05556 2/20 0.42
ITGA4 P13612 2/20 0.42
SMO Q99835 1/20 0.40
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPK1 P28482 1/20 0.38
ADRB1 P08588 8/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ADRB2 P07550 2/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6540024 1.00 BACE1 (0.53) BACE1ADRB3ITGB1ITGA4SMO
SCHEMBL6539651 0.89 ADRB3 (0.47) BACE1ADRB3SMOADRB1ADRB2
SCHEMBL6539659 0.89 ADRB3 (0.47) BACE1ADRB3SMOADRB1ADRB2
SCHEMBL6539237 0.82 BACE1 (0.52) BACE1ADRB3ITGB1ITGA4ADRB1
SCHEMBL6539232 0.82 BACE1 (0.52) BACE1ADRB3ITGB1ITGA4ADRB1
SCHEMBL6539195 0.79 BACE1 (0.54) BACE1ADRB3ADRB1ADRB2ADRA1D
SCHEMBL6538940 0.79 BACE1 (0.54) BACE1ADRB3ADRB1ADRB2ADRA1D
SCHEMBL6538935 0.79 BACE1 (0.54) BACE1ADRB3ADRB1ADRB2ADRA1D
SCHEMBL6478726 0.74 BACE1 (0.52) BACE1ADRB3ADRB1ADRB2ADRA1D
SCHEMBL6478721 0.74 BACE1 (0.52) BACE1ADRB3ADRB1ADRB2ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6826033-B2 BETA 3 ADRENERGIC RECEPTOR AGONISTS; TREATMENT OF POLLAKIURIA, URINARY INCONTINENCE, OBESITY OR DIABETES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-11-30 US disclosed
US-20040037022-A1 Aminoalcohol derivatives ASTELLAS PHARMA INC. (JP) 2004-02-26 US disclosed