SCHEMBL6540648

SCHEMBL6540648

C[C@H](Cc1ccc(S(=O)(=O)c2ccc(O)c(Cl)c2)cc1)NC(=O)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.41
ACACB O00763 5/20 0.40
PDK1 Q15118 5/20 0.39
PDK2 Q15119 5/20 0.39
PDK3 Q15120 5/20 0.39
PDK4 Q16654 5/20 0.39
CNR1 P21554 2/20 0.39
ESR1 P03372 1/20 0.39
KCNH2 Q12809 1/20 0.39
ABCC9 O60706 2/20 0.38
ABCC8 Q09428 2/20 0.38
KCNJ11 Q14654 2/20 0.38
KCNJ8 Q15842 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6810020 1.00 ABCB11 (0.41) ABCB11ACACBPDK1PDK2PDK3
SCHEMBL6540415 0.88 CNR1 (0.40) ACACBCNR1ESR1KCNH2ABCC9
SCHEMBL6540853 0.88 ESR1 (0.42) ACACBCNR1ESR1KCNH2ABCC9
SCHEMBL6540590 0.86 ACACB (0.45) ACACBPDK1PDK2PDK3PDK4
SCHEMBL6806001 0.86 ACACB (0.45) ACACBPDK1PDK2PDK3PDK4
SCHEMBL6677754 0.86 ALDH1A1 (0.42) ACACBCNR1ESR1KCNH2GAA
SCHEMBL6800681 0.86 ALDH1A1 (0.42) ACACBCNR1ESR1KCNH2GAA
SCHEMBL6541437 0.85 ESR1 (0.46) ACACBCNR1ESR1KCNH2ABCC9
SCHEMBL6539913 0.85 ESR1 (0.46) ACACBCNR1ESR1KCNH2ABCC9
SCHEMBL6805794 0.84 MAPT (0.42) ACACBCNR1ESR1KCNH2ABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040138462-A1 Aminoalcohol derivatives ASTELLAS PHARMA INC. (JP) 2004-07-15 US disclosed
US-20040106653-A1 Aminoalcohol derivatives FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-06-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040138462-A1 Aminoalcohol derivatives BPHL, FANCD2, HRH2 ABCB11 1184/4885ACACB 3020/4885PDK1 2885/4885
US-20040106653-A1 Aminoalcohol derivatives FANCD2, FANCI, HRH2 ABCB11 1249/4885ACACB 1800/4885PDK1 3748/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.