SCHEMBL654460

SCHEMBL654460

O=C(O)N1C[C@H]2N(c3cnc(Cl)c(Cl)c3)C[C@@]2(Cc2ccccc2)C1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CHRNB2 P17787 8/20 0.40
CHRNA4 P43681 8/20 0.40
CHRNB4 P30926 6/20 0.36
CHRNA3 P32297 6/20 0.36
ALDH1A1 P00352 4/20 0.36
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GRIN2B Q13224 2/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
SCD5 Q86SK9 1/20 0.32
EPHX2 P34913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL652521 0.90 CHRNB2 (0.42) MEN1KMT2ACHRNB2CHRNA4CHRNB4
SCHEMBL653486 0.85 GRIN2B (0.42) CHRNB2CHRNA4CHRNB4CHRNA3ALDH1A1
SCHEMBL649307 0.85 GRIN2B (0.42) CHRNB2CHRNA4CHRNB4CHRNA3ALDH1A1
SCHEMBL654323 0.85 GRIN2B (0.42) CHRNB2CHRNA4CHRNB4CHRNA3ALDH1A1
SCHEMBL650794 0.80 SMN1; SMN2 (0.37) CHRNB2CHRNA4CHRNB4CHRNA3ALDH1A1
SCHEMBL653615 0.80 SMN1; SMN2 (0.37) CHRNB2CHRNA4CHRNB4CHRNA3ALDH1A1
SCHEMBL653675 0.80 CHRNB2 (0.41) MEN1KMT2ACHRNB2CHRNA4CHRNB4
SCHEMBL929834 0.80 CHRNB2 (0.41) CHRNB2CHRNA4CHRNB4CHRNA3ALDH1A1
SCHEMBL651156 0.79 ARG1 (0.39) MEN1KMT2ACHRNB2CHRNA4CHRNB4
SCHEMBL651858 0.79 ARG1 (0.39) MEN1KMT2ACHRNB2CHRNA4CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119635-B2 Diazabicyclic central nervous system active agents ABBOTT LABORATORIES (US) 2012-02-21 US disclosed
EP-2298775-A1 Diazabicyclic central nervous system active agents Abbott Laboratories (US) 2011-03-23 EP disclosed
EP-2295437-A1 Diazabicyclic central nervous system active agents Abbott Laboratories (US) 2011-03-16 EP disclosed