SCHEMBL6544836

SCHEMBL6544836

Cc1cc(Oc2ccc(N)c(N(C)C(=O)O)c2)ccc1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 7/20 0.38
THRA P10827 6/20 0.38
PDE10A Q9Y233 1/20 0.37
ESR1 P03372 2/20 0.35
AR P10275 1/20 0.35
ESR2 Q92731 1/20 0.35
ESRRA P11474 1/20 0.35
HSD17B1 P14061 1/20 0.35
HSD17B2 P37059 1/20 0.35
NR4A1 P22736 1/20 0.35
PCNA P12004 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
RECQL P46063 1/20 0.33
BLM P54132 1/20 0.33
KMT2A Q03164 1/20 0.33
MCL1 Q07820 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3488405 0.89 TDP1 (0.42) ESR1ESR2HSD17B1HSD17B2NR4A1
SCHEMBL3487567 0.85 CHEK2 (0.39) HSD17B1HSD17B2NR4A1
SCHEMBL6543782 0.85 PARP10 (0.42) THRBTHRAESR1ESR2NR4A1
SCHEMBL3488177 0.85 HSD17B1 (0.44) HSD17B1HSD17B2NR4A1ALDH1A1MAPT
SCHEMBL6543660 0.84 ESRRA (0.37) THRBTHRAPDE10AESR1AR
SCHEMBL3487710 0.83 MRGPRX4 (0.38) HSD17B1HSD17B2NR4A1KMT2A
SCHEMBL3488383 0.82 PARP10 (0.45) HSD17B1HSD17B2NR4A1MEN1KMT2A
SCHEMBL3488037 0.82 ALDH1A1 (0.39) ARNR4A1MEN1ALDH1A1GAA
SCHEMBL3487215 0.81 HSD17B1 (0.52) HSD17B1HSD17B2MEN1ALDH1A1GAA
SCHEMBL3488333 0.81 BRAF (0.44) MEN1ALDH1A1MAPTBLMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1022272-B1 SUBSTITUTED FUSED HETEROCYCLIC COMPOUNDS SANKYO CO (JP) 2004-05-26 EP disclosed
US-6432993-B1 BENZIMIDAZOLE OR IMIDAZO(4,5-B)PYRIDINE DERIVATES; IMMUNOMODULATORS; ALDOSE REDUCTASE AND LIPOXYGENASE INHIBITORS; DIABETES; PREVENTS LIPID PEROXIDATION; ANTILIPEMIC, HYPOTENSIVE AGENTS SANKYO COMPANY, LIMITED (JP) 2002-08-13 US disclosed
EP-1022272-A1 SUBSTITUTED FUSED HETEROCYCLIC COMPOUNDS Sankyo Company Limited (JP) 2000-07-26 EP disclosed