SCHEMBL6545762

SCHEMBL6545762

CC(=O)Nc1nc(-c2ccncc2)c(-c2ccc(C(C)(C)C)cc2)s1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.62
MAPT P10636 2/20 0.62
KDM4E B2RXH2 2/20 0.62
LMNA P02545 1/20 0.62
GAA P10253 1/20 0.62
ADORA3 P0DMS8 8/20 0.60
ADORA2B P29275 3/20 0.60
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
ADORA1 P30542 6/20 0.49
ADORA2A P29274 5/20 0.49
PIK3CD O00329 3/20 0.47
PIK3CA P42336 3/20 0.47
PIK3CB P42338 3/20 0.47
PIK3CG P48736 3/20 0.47
CHRM5 P08912 1/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
KIF11 P52732 1/20 0.45
XIAP P98170 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6278341 1.00 ALDH1A1 (0.62) ALDH1A1MAPTKDM4ELMNAGAA
SCHEMBL6546759 0.90 ALDH1A1 (0.62) ALDH1A1MAPTKDM4ELMNAGAA
SCHEMBL6545850 0.87 XIAP (0.53) ALDH1A1MAPTKDM4ELMNAGAA
SCHEMBL6546289 0.87 KDM4E (0.51) ALDH1A1MAPTKDM4ELMNAGAA
SCHEMBL6546864 0.87 KDM4E (0.51) ALDH1A1MAPTKDM4ELMNAGAA
SCHEMBL6282412 0.86 ADORA1 (0.59) ALDH1A1MAPTKDM4ELMNAADORA3
SCHEMBL6545559 0.86 ALDH1A1 (0.56) ALDH1A1MAPTKDM4ELMNAGAA
Hydrochloric Acid SCHEMBL6618039 0.85 ADORA3 (0.45) ALDH1A1MAPTKDM4ELMNAGAA
SCHEMBL6546278 0.85 ABL1 (0.54) ALDH1A1MAPTKDM4ELMNAGAA
SCHEMBL6546272 0.85 ALDH1A1 (0.50) ALDH1A1MAPTKDM4ELMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1027050-B1 1,3-THIAZOLES AS ADENOSINE A3 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF ALLERGY, ASTHMA AND DIABETES TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-01-14 EP disclosed
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed