SCHEMBL6545801

SCHEMBL6545801

C=CCOC(=O)C(C=O)=[N+]=[N-]

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.35
TSHR P16473 2/20 0.33
MAPT P10636 1/20 0.33
CACNA1B Q00975 1/20 0.33
APBA1 Q02410 1/20 0.33
ALDH1A1 P00352 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8970712 0.78 CYP3A4 (0.38) CYP3A4TSHRMAPTCACNA1BAPBA1
SCHEMBL71162 0.76 NPSR1 (0.41) TSHRMAPTALDH1A1HSD17B10
SCHEMBL177943 0.73 CYP3A4 (0.48) CYP3A4TSHRMAPTCACNA1BAPBA1
SCHEMBL2541412 0.73 CYP3A4 (0.35) CYP3A4TSHRMAPTCACNA1BAPBA1
SCHEMBL27807560 0.73 CYP3A4 (0.41) CYP3A4TSHRMAPTCACNA1BAPBA1
SCHEMBL8409550 0.72 CYP3A4 (0.43) CYP3A4TSHRMAPTCACNA1BAPBA1
SCHEMBL9167074 0.72 TSHR (0.36) CYP3A4TSHRMAPTCACNA1BAPBA1
SCHEMBL7512684 0.71 CYP3A4 (0.46) CYP3A4TSHRMAPTCACNA1BAPBA1
SCHEMBL10966895 0.69 CYP3A4 (0.45) CYP3A4TSHRMAPTCACNA1BAPBA1
SCHEMBL21980975 0.69 CYP3A4 (0.45) CYP3A4TSHRMAPTCACNA1BAPBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1250330-B1 PROCESS FOR THE PREPARATION OF 3-FUROATE ESTERS AND NOVEL INTERMEDIATE COMPOUNDS EASTMAN CHEM CO (US) 2004-01-07 EP disclosed
EP-1250330-A1 PROCESS FOR THE PREPARATION OF 3-FUROATE ESTERS AND NOVEL INTERMEDIATE COMPOUNDS EASTMAN CHEMICAL COMPANY (US) 2002-10-23 EP disclosed
WO-2001055127-A1 PROCESS FOR THE PREPARATION OF 3-FUROATE ESTERS AND NOVEL INTERMEDIATE COMPOUNDS EASTMAN CHEMICAL COMPANY (US) 2001-08-02 WO disclosed
US-6184394-B1 ALKYL 3-FUROATES FROM 4-ACYL-2,3-DIHYDROFURANS FROM 4-ACYL-2,3-DIHYDRO-FURANS BY HALOGENATING IN THE PRESENCE OF AN ALKANOL FOLLOWED BY CONTACTING WITH A STRONG BASE; DRUGS; ANTINFLAMMATORY AND -FOULING AGENTS EASTMAN CHEMICAL COMPANY 2001-02-06 US disclosed