SCHEMBL6545950

SCHEMBL6545950

N#CC(C(=O)c1cccnc1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
APP P05067 1/20 0.50
GAA P10253 1/20 0.50
HCAR3 P49019 1/20 0.50
HCAR2 Q8TDS4 1/20 0.50
HTT P42858 1/20 0.49
EPHX2 P34913 2/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
PLOD2 O00469 1/20 0.47
LMNA P02545 1/20 0.45
F7 P08709 1/20 0.45
F3 P13726 1/20 0.45
SARM1 Q6SZW1 1/20 0.45
SIRT2 Q8IXJ6 1/20 0.45
SIRT6 Q8N6T7 1/20 0.45
SIRT1 Q96EB6 1/20 0.45
SIRT3 Q9NTG7 1/20 0.45
SIRT5 Q9NXA8 1/20 0.45
SIRT4 Q9Y6E7 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4328721 0.87 MAPT (0.47) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL5505530 0.84 L3MBTL1 (0.61) ALDH1A1HTTLMNAPOLB
SCHEMBL14519387 0.83 L3MBTL1 (0.49) ALDH1A1CYP2C9CYP2C19PLOD2LMNA
SCHEMBL838079 0.83 L3MBTL1 (0.52) ALDH1A1HTTEPHX2CYP2C9CYP2C19
SCHEMBL7202862 0.80 L3MBTL1 (0.55) ALDH1A1HTTLMNA
SCHEMBL7200938 0.79 TDP1 (0.50) ALDH1A1HTTLMNAPOLB
SCHEMBL27380660 0.78 POLB (0.48) ALDH1A1HTTEPHX2LMNAPOLB
SCHEMBL8836116 0.78 POLB (0.48) ALDH1A1HTTEPHX2LMNAPOLB
SCHEMBL10880279 0.78 SMN1; SMN2 (0.52) ALDH1A1GAAHTTLMNAPOLB
SCHEMBL2582102 0.78 ALDH1A1 (0.52) ALDH1A1APPGAAHCAR3HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1027050-B1 1,3-THIAZOLES AS ADENOSINE A3 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF ALLERGY, ASTHMA AND DIABETES TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-01-14 EP disclosed
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed
EP-0046451-A2 Diaryl-imidazole compounds, methods for their preparation, pharmaceutical drugs containing them and their use CIBA-GEIGY AG (CH) 1982-02-24 EP disclosed