SCHEMBL654702

SCHEMBL654702

c1ccc([C](c2ccccc2)c2ccc(NC(c3ccccc3)(c3ccccc3)c3ccccc3)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 2/20 0.42
MAPK12 P53778 2/20 0.42
MAPK11 Q15759 2/20 0.42
MAPK14 Q16539 2/20 0.42
RAB9A P51151 4/20 0.40
NPC1 O15118 2/20 0.40
KCNN4 O15554 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 5/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
FFAR1 O14842 1/20 0.37
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 3/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PTPN1 P18031 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11279906 0.80 KCNN4 (0.52) KCNN4MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL23112981 0.75 KCNN4 (0.43) KCNN4ALDH1A1L3MBTL1
SCHEMBL18035826 0.75 ALDH1A1 (0.44) RAB9ANPC1KCNN4MEN1KMT2A
Biphenyl SCHEMBL7519251 0.72 KCNN4 (0.44) KCNN4ALDH1A1L3MBTL1LMNA
SCHEMBL14855117 0.72 IDO1 (0.62) MAPK13MAPK12MAPK11MAPK14RAB9A
SCHEMBL8177 0.72 CES1 (0.40) RAB9ANPC1KCNN4ALDH1A1L3MBTL1
SCHEMBL574740 0.71 CA1 (0.57) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL874147 0.71 KCNN4 (0.43) KCNN4ALDH1A1VNN1HDAC3HDAC4
SCHEMBL7535593 0.71 KCNN4 (0.39) RAB9AKCNN4MEN1KMT2AALDH1A1
SCHEMBL11586969 0.71 AKR1B1 (0.53) RAB9AMEN1KMT2AALDH1A1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119657-B2 Enantiomeric compositions of 2-amino-1-(2-isopropylpyrazolo[1,5-α]pyridin-3-yl)propan-1-one and related methods MEDICINOVA, INC. (US) 2012-02-21 US disclosed