SCHEMBL6548458

SCHEMBL6548458

O=c1c2[nH]cnc2ncn1Cc1ccc2ccccc2c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.50
GAA P10253 1/20 0.41
DAO P14920 1/20 0.40
SIRT2 Q8IXJ6 4/20 0.40
CDC7 O00311 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP19A1 P11511 1/20 0.40
ACP1 P24666 2/20 0.40
PDE10A Q9Y233 1/20 0.39
ADORA2A P29274 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3306010 0.84 ACP1 (0.55) TRPA1LMNAHPGDSMN1; SMN2ACP1
SCHEMBL6548460 0.82 DAO (0.43) TRPA1GAADAOALDH1A1LMNA
Bromide SCHEMBL6556197 0.79 SIRT2 (0.41) TRPA1GAADAOSIRT2CYP19A1
SCHEMBL4966803 0.78 PNP (0.50) ALDH1A1POLBSMN1; SMN2
Hydrochloric Acid SCHEMBL25426121 0.77 PNP (0.49) ALDH1A1POLBSMN1; SMN2
SCHEMBL7120147 0.75 DAO (0.40) TRPA1GAADAOSIRT2ALDH1A1
SCHEMBL8509077 0.72 SMN1; SMN2 (0.47) TRPA1ALDH1A1LMNAMAPTHPGD
SCHEMBL6797064 0.71 GAA (0.43) TRPA1GAASIRT2ALDH1A1POLB
SCHEMBL7111737 0.71 PNP (0.49) TRPA1DAOALDH1A1HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL6258586 0.70 PNP (0.48) TRPA1DAOALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383766-A1 DISUBSTITUTED 1,7-GUANINES Pharmacia Italia S.p.A. (IT) 2004-01-28 EP claimed
WO-2002090357-A1 DISUBSTITUTED 1,7-GUANINES PHARMACIA ITALIA S.P.A. (IT) 2002-11-14 WO claimed
EP-1383766-A1 DISUBSTITUTED 1,7-GUANINES Pharmacia Italia S.p.A. (IT) 2004-01-28 EP disclosed
WO-2002090357-A1 DISUBSTITUTED 1,7-GUANINES PHARMACIA ITALIA S.P.A. (IT) 2002-11-14 WO disclosed