SCHEMBL6548460

SCHEMBL6548460

O=c1[nH]cnc2ncn(Cc3ccc4ccccc4c3)c12

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.43
TRPA1 O75762 1/20 0.43
SMN1; SMN2 Q16637 4/20 0.42
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 2/20 0.42
HPGD P15428 1/20 0.40
CYP19A1 P11511 1/20 0.40
PDE10A Q9Y233 1/20 0.39
GAA P10253 2/20 0.38
ADORA2A P29274 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
ACHE P22303 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2958439 0.84 SMN1; SMN2 (0.53) SMN1; SMN2ALDH1A1KMT2AHPGD
SCHEMBL6548458 0.82 TRPA1 (0.50) DAOTRPA1SMN1; SMN2ALDH1A1HPGD
SCHEMBL7111737 0.81 PNP (0.49) DAOTRPA1SMN1; SMN2ALDH1A1KMT2A
SCHEMBL7120147 0.80 DAO (0.40) DAOTRPA1SMN1; SMN2ALDH1A1KMT2A
Hydrochloric Acid SCHEMBL6258586 0.80 PNP (0.48) DAOTRPA1SMN1; SMN2ALDH1A1KMT2A
SCHEMBL7985648 0.79 HPGD (0.47) DAOTRPA1SMN1; SMN2ALDH1A1KMT2A
SCHEMBL20187449 0.79 QPCTL (0.47) TRPA1ALDH1A1KMT2AHPGDGAA
SCHEMBL22533556 0.76 KMT2A (0.41) TRPA1SMN1; SMN2ALDH1A1KMT2AHPGD
SCHEMBL27441619 0.76 KMT2A (0.41) TRPA1SMN1; SMN2ALDH1A1KMT2AHPGD
Bromide SCHEMBL6556197 0.74 SIRT2 (0.41) DAOTRPA1CYP19A1PDE10AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383766-A1 DISUBSTITUTED 1,7-GUANINES Pharmacia Italia S.p.A. (IT) 2004-01-28 EP claimed
WO-2002090357-A1 DISUBSTITUTED 1,7-GUANINES PHARMACIA ITALIA S.P.A. (IT) 2002-11-14 WO claimed
EP-1383766-A1 DISUBSTITUTED 1,7-GUANINES Pharmacia Italia S.p.A. (IT) 2004-01-28 EP disclosed
WO-2002090357-A1 DISUBSTITUTED 1,7-GUANINES PHARMACIA ITALIA S.P.A. (IT) 2002-11-14 WO disclosed