SCHEMBL6548684

SCHEMBL6548684

COc1ccc(N=C(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.55
HTR3E A5X5Y0 1/20 0.55
HTR3B O95264 1/20 0.55
HTR3A P46098 1/20 0.55
HTR3D Q70Z44 1/20 0.55
HTR3C Q8WXA8 1/20 0.55
CES2 O00748 1/20 0.53
CES1 P23141 1/20 0.53
ESR1 P03372 3/20 0.53
ESR2 Q92731 3/20 0.53
CA4 P22748 1/20 0.48
MGLL Q99685 1/20 0.48
LTA4H P09960 1/20 0.47
MAPT P10636 4/20 0.47
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPK1 P28482 2/20 0.47
GAA P10253 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19505630 0.92 ESR1 (0.60) NOS3HTR3EHTR3BHTR3AHTR3D
SCHEMBL17017261 0.92 ESR2 (0.66) NOS3HTR3EHTR3BHTR3AHTR3D
SCHEMBL24105688 0.90 ESR2 (0.61) NOS3HTR3EHTR3BHTR3AHTR3D
SCHEMBL30951898 0.88 ESR2 (0.59) NOS3HTR3EHTR3BHTR3AHTR3D
SCHEMBL5608124 0.83 NPC1 (0.51) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL12629405 0.83 NOS3 (0.58) NOS3HTR3EHTR3BHTR3AHTR3D
SCHEMBL3179816 0.83 NOS3 (0.58) NOS3HTR3EHTR3BHTR3AHTR3D
SCHEMBL15136973 0.83 NOS3 (0.58) NOS3HTR3EHTR3BHTR3AHTR3D
SCHEMBL11522898 0.81 NOS3 (0.52) NOS3HTR3EHTR3BHTR3AHTR3D
SCHEMBL8815637 0.81 NOS3 (0.52) NOS3HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130253185-A1 NOVEL CATALYSTS DALHOUSIE UNIVERSITY (CA) 2013-09-26 US disclosed
EP-1100774-B1 IMPROVED ARYLAMINE SYNTHESIS MASSACHUSETTS INST TECHNOLOGY (US) 2004-01-21 EP disclosed
US-6323366-B1 ACTIVATED ARYL GROUP AND AN IMINE GROUP ARE COMBINED, IN THE PRESENCE OF A TRANSITION METAL CATALYST FOR FORMATION OF A CARBON-NITROGEN BOND BETWEEN THE ACTIVATED CARBON OF THE ARENE AND IMINE NITROGEN; CONVERTING TO ARYLAMINE MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2001-11-27 US disclosed
EP-1100774-A1 IMPROVED ARYLAMINE SYNTHESIS MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2001-05-23 EP disclosed
WO-2000005199-A1 IMPROVED ARYLAMINE SYNTHESIS MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2000-02-03 WO disclosed