SCHEMBL5608124

SCHEMBL5608124

COc1cc(N=C(c2ccccc2)c2ccccc2)cc(OC)c1

nearest known ligand 0.90

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
HTT P42858 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
ALDH1A1 P00352 2/20 0.44
GAA P10253 1/20 0.44
ESR1 P03372 2/20 0.44
ESR2 Q92731 2/20 0.44
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
MGLL Q99685 1/20 0.43
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6547586 0.86 HTR3E (0.62) NPC1RAB9AHTTSMN1; SMN2ESR1
SCHEMBL6548684 0.83 NOS3 (0.55) NPC1RAB9ASMN1; SMN2ALDH1A1GAA
SCHEMBL19505630 0.79 ESR1 (0.60) NPC1RAB9ASMN1; SMN2ALDH1A1GAA
SCHEMBL17017261 0.76 ESR2 (0.66) ESR1ESR2HTR3EHTR3BHTR3A
SCHEMBL5604475 0.75 ESR2 (0.53) HTTSMN1; SMN2ALDH1A1GAAESR1
SCHEMBL12809830 0.74 CDC25B (0.46) NPC1RAB9AHTTSMN1; SMN2PDE4A
SCHEMBL30305252 0.74 CDC25B (0.46) NPC1RAB9AHTTSMN1; SMN2PDE4A
SCHEMBL24451315 0.73 ESR1 (0.68) NPC1RAB9AHTTPDE4APDE4D
SCHEMBL31229397 0.73 ATP4A (0.41) NPC1RAB9AHTTSMN1; SMN2PDE4A
SCHEMBL4450591 0.73 ESR2 (0.74) ALDH1A1ESR1ESR2HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1354887-B1 Ligands for metals and improved metal-catalyzed processes based thereon MASSACHUSETTS INST TECHNOLOGY (US) 2007-04-25 EP disclosed
EP-1097158-B1 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INST TECHNOLOGY (US) 2006-01-25 EP disclosed
EP-1100774-B1 IMPROVED ARYLAMINE SYNTHESIS MASSACHUSETTS INST TECHNOLOGY (US) 2004-01-21 EP disclosed
EP-1354887-A1 Ligands for metals and improved metal-catalyzed processes based thereon Massachusetts Insitute of Technology (US) 2003-10-22 EP disclosed
EP-1097158-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2001-05-09 EP disclosed
WO-2000002887-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2000-01-20 WO disclosed