SCHEMBL6549005

SCHEMBL6549005

COc1ccc(S(=O)(=O)C#C[Si](C)(C)C)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 4/20 0.53
GAA P10253 1/20 0.50
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
MMP2 P08253 2/20 0.46
MMP8 P22894 2/20 0.46
MMP13 P45452 2/20 0.46
MMP1 P03956 1/20 0.46
MMP9 P14780 1/20 0.46
NPC1 O15118 1/20 0.44
PKLR P30613 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 2/20 0.42
PTGS2 P35354 1/20 0.42
F2 P00734 1/20 0.42
PRSS1 P07477 1/20 0.42
PRSS2 P07478 1/20 0.42
PRSS3 P35030 1/20 0.42
CA9 Q16790 2/20 0.41
RAPGEF4 Q8WZA2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6547655 0.79 PKM (0.55) PKMGAACA1CA2MMP2
SCHEMBL28442170 0.78 PKM (0.53) PKMGAACA1CA2MMP2
Anisole SCHEMBL7455194 0.76 CA4 (0.50) PKMGAANPC1RAB9AALDH1A1
SCHEMBL4388431 0.76 ALDH1A1 (0.44) CA1CA2MMP2MMP8MMP13
SCHEMBL8080302 0.76 ALDH1A1 (0.44) CA1CA2MMP2MMP8MMP13
SCHEMBL10746956 0.75 PKM (0.59) PKMGAACA1CA2MMP2
SCHEMBL6549282 0.75 PKM (0.59) PKMGAACA1CA2MMP2
SCHEMBL28281705 0.74 NPC1 (0.50) PKMGAACA1CA2MMP2
SCHEMBL28440362 0.73 CA12 (0.49) PKMGAACA1CA2NPC1
SCHEMBL31619031 0.71 MEN1 (0.47) PKMGAANPC1PKLRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1162962-B1 ALKYNYL ARYL SULFONES LONZA AG (US) 2004-12-01 EP disclosed
EP-1162962-A4 ALKYNYL ARYL SULFONES LONZA AG (US) 2002-10-30 EP disclosed
EP-1162962-A1 ALKYNYL ARYL SULFONES LONZA INC. (US) 2001-12-19 EP disclosed
US-6232503-B1 MICROBIOCIDES LONZA INC. 2001-05-15 US disclosed
WO-2000056305-A1 ALKYNYL ARYL SULFONES LONZA INC. (US) 2000-09-28 WO disclosed