SCHEMBL6552293

SCHEMBL6552293

CC(C)(Sc1ccc(CCNC(=O)OCC2c3ccccc3-c3ccccc32)cc1)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.52
OPRD1 P41143 1/20 0.41
PPARG P37231 4/20 0.41
PPARA Q07869 4/20 0.41
PPARD Q03181 2/20 0.41
EPHX2 P34913 1/20 0.40
MDM4 O15151 1/20 0.40
TP53 P04637 1/20 0.40
CASP3 P42574 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7871514 0.89 KMT2A (0.47) KMT2AOPRD1EPHX2CASP3
SCHEMBL6032374 0.83 KMT2A (0.67) KMT2AOPRD1EPHX2CASP3HDAC3
SCHEMBL30570803 0.80 KMT2A (0.63) KMT2AOPRD1EPHX2CASP3HDAC3
SCHEMBL14247589 0.80 KMT2A (0.60) KMT2AOPRD1EPHX2CASP3HDAC3
SCHEMBL18740102 0.80 KMT2A (0.63) KMT2AOPRD1EPHX2CASP3HDAC3
SCHEMBL2416313 0.79 KMT2A (0.47) KMT2AEPHX2MDM4TP53CASP3
SCHEMBL15434605 0.77 KMT2A (0.61) KMT2AEPHX2MDM4TP53CASP3
SCHEMBL15548985 0.75 KMT2A (0.66) KMT2AOPRD1HDAC3HDAC4HDAC1
SCHEMBL15726427 0.75 KMT2A (0.62) KMT2AEPHX2MDM4TP53CASP3
SCHEMBL23270799 0.75 KMT2A (0.62) KMT2AOPRD1EPHX2HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1149063-B1 UREIDO-THIOBUTYRIC ACID DERIVATIVES AS PPAR-AGONISTS SMITHKLINE BEECHAM CORP (US) 2004-12-15 EP disclosed
EP-1149063-A2 UREIDO-THIOBUTYRIC ACID DERIVATIVES AS PPAR-AGONISTS GLAXO GROUP LIMITED (GB) 2001-10-31 EP disclosed
WO-2000023407-A2 UREIDO-THIOBUTYRIC ACID DERIVATIVES AS PPAR-AGONISTS GLAXO GROUP LIMITED (GB) 2000-04-27 WO disclosed