SCHEMBL6555370

SCHEMBL6555370

O=C(Nc1cc(Br)ccc1CCN1CCOCC1)C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.44
MAPT P10636 3/20 0.43
ALDH1A1 P00352 5/20 0.43
KMT2A Q03164 4/20 0.43
MPI P34949 1/20 0.43
ABL1 P00519 1/20 0.42
RIN1 Q13671 1/20 0.42
TSHR P16473 3/20 0.42
HTT P42858 2/20 0.42
CNR2 P34972 2/20 0.41
MEN1 O00255 2/20 0.40
ALOX12 P18054 1/20 0.40
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6555185 0.88 CNR2 (0.47) LMNAMAPTALDH1A1KMT2ATSHR
SCHEMBL17351215 0.75 MAPT (0.36) LMNAMAPTKMT2AHTTMEN1
SCHEMBL15137221 0.73 TSHR (0.47) LMNAMAPTALDH1A1KMT2AMPI
SCHEMBL6557378 0.73 CYP1A2 (0.38) LMNAMAPTALDH1A1ALOX12
SCHEMBL27857544 0.71 CYP2A13 (0.46) LMNAMAPTALDH1A1KMT2AMPI
SCHEMBL27496539 0.70 SLC6A4 (0.41) LMNAMAPTKMT2AMEN1
SCHEMBL1977685 0.70 CYP2A13 (0.51) LMNAMAPTALDH1A1KMT2AHTT
SCHEMBL4189779 0.69 CSF1R (0.67)
SCHEMBL445310 0.69 ALDH1A1 (0.60) LMNAALDH1A1
SCHEMBL6866035 0.68 SLC6A2 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230224-B1 SUBSTITUTED 5-BENZYL-2,4-DIAMINOPYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2004-12-29 EP disclosed
US-6821980-B1 Substituted 5-benzyl-2,4-diaminopyrimidines BASILEA PHARMACEUTICA AG (CH) 2004-11-23 US disclosed
EP-1230224-A1 SUBSTITUTED 5-BENZYL-2,4-DIAMINOPYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 2002-08-14 EP disclosed
WO-2001032633-A1 SUBSTITUTED 5-BENZYL-2,4-DIAMINOPYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2001-05-10 WO disclosed