SCHEMBL6555963

SCHEMBL6555963

O=c1[nH]c2ccc(CCCC3CC(c4ccc(C(F)(F)F)cc4)=CCN3)cc2c2ccc(Cl)cc12

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.39
CYP2C9 P11712 6/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
CTSC P53634 2/20 0.36
RAD51 Q06609 1/20 0.36
CNR1 P21554 2/20 0.33
PGR P06401 1/20 0.33
SNCA P37840 1/20 0.33
OPRM1 P35372 1/20 0.33
CTSK P43235 1/20 0.32
CDC25A P30304 1/20 0.32
CDC25C P30307 1/20 0.32
TNKS O95271 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6409099 0.79 PARP1 (0.65) PARP1
SCHEMBL6555513 0.77 PARP1 (0.59) PARP1CYP1A2TNKS
Hydrochloric Acid SCHEMBL6554106 0.72 PARP1 (0.40) PARP1
SCHEMBL6555511 0.70 PARP1 (0.54) PARP1CYP1A2CTSCCDC25ACDC25C
SCHEMBL6410344 0.69 PARP1 (0.68) PARP1
SCHEMBL6554152 0.67 PARP1 (0.38) PARP1
SCHEMBL8542783 0.64 MAOB (0.42)
SCHEMBL20227575 0.64 SIRT1 (0.47) PARP1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL7439313 0.62 MAOB (0.46)
SCHEMBL19857834 0.61 MAP2 (0.53) CYP2C9CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487800-A1 PHENANTHRIDINONES AS PARP INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-12-22 EP disclosed
WO-2003080581-A1 PHENANTHRIDINONES AS PARP INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-10-02 WO disclosed