SCHEMBL6558462

SCHEMBL6558462

COc1ccc2c(c1)C(=O)C[C@H]1CN(C)C[C@@H]21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP19A1 P11511 5/20 0.41
SIGMAR1 Q99720 2/20 0.41
MAP2K3 P46734 1/20 0.41
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
ACHE P22303 1/20 0.40
ABCB1 P08183 1/20 0.40
AR P10275 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
BRD4 O60885 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6558458 1.00 KDM4E (0.42) KDM4EALDH1A1GAAMAPTALOX15
SCHEMBL6558466 1.00 KDM4E (0.42) KDM4EALDH1A1GAAMAPTALOX15
Fumaric Acid SCHEMBL6556397 0.91 KMT2A (0.40) KDM4EALDH1A1GAAMAPTALOX15
Fumaric Acid SCHEMBL6556402 0.91 KMT2A (0.40) KDM4EALDH1A1GAAMAPTALOX15
Fumaric Acid SCHEMBL6556387 0.91 KMT2A (0.40) KDM4EALDH1A1GAAMAPTALOX15
Fumaric Acid SCHEMBL6556392 0.91 KMT2A (0.40) KDM4EALDH1A1GAAMAPTALOX15
SCHEMBL6556481 0.89 GAA (0.45) KDM4EALDH1A1GAAMAPTALOX15
SCHEMBL6556478 0.89 GAA (0.45) KDM4EALDH1A1GAAMAPTALOX15
SCHEMBL6556471 0.89 GAA (0.45) KDM4EALDH1A1GAAMAPTALOX15
SCHEMBL6556584 0.88 SIGMAR1 (0.47) KDM4EALDH1A1MAPTALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6310208-B1 Serotonin receptor binding benzo[e]isoindoles and benzo[h]isoquinolines HOFFMANN-LA ROCHE INC. 2001-10-30 US claimed
EP-0958285-B1 TRICYCLIC BENZO[e]ISOINDOLES AND BENZO[h]ISOQUINOLINES HOFFMANN LA ROCHE (CH) 2004-01-07 EP disclosed
US-6310208-B1 Serotonin receptor binding benzo[e]isoindoles and benzo[h]isoquinolines HOFFMANN-LA ROCHE INC. 2001-10-30 US disclosed