SCHEMBL6559364

SCHEMBL6559364

Nc1cccc(C(=O)Nc2ccc(C(F)(F)F)cc2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 7/20 1.00
NPC1 O15118 2/20 0.69
RAB9A P51151 2/20 0.69
LMNA P02545 2/20 0.62
MAPT P10636 2/20 0.60
KCNK3 O14649 1/20 0.59
P2RX1 P51575 2/20 0.58
TRPV1 Q8NER1 2/20 0.57
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
EPHX2 P34913 1/20 0.57
RHOC P08134 1/20 0.56
RHOA P61586 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2127722 0.87 PTGS1 (0.77) PTGS1NPC1RAB9ALMNAMAPT
SCHEMBL4463935 0.87 PTGS1 (0.89) PTGS1RAB9ALMNAMAPTKCNK3
SCHEMBL548237 0.86 PTGS1 (0.77) PTGS1NPC1RAB9ALMNAMAPT
SCHEMBL11593046 0.86 PTGS1 (0.75) PTGS1NPC1RAB9ALMNAMAPT
SCHEMBL3454009 0.85 PTGS1 (1.00) PTGS1NPC1RAB9ALMNAMAPT
SCHEMBL17744815 0.84 KMT2A (0.73) PTGS1LMNAMAPTMEN1KMT2A
SCHEMBL309467 0.84 PTGS1 (0.72) PTGS1LMNAMAPTMEN1KMT2A
SCHEMBL31171945 0.84 PTGS1 (0.72) PTGS1LMNAMAPTMEN1KMT2A
SCHEMBL2861430 0.84 PTGS1 (1.00) PTGS1RAB9ALMNAMAPTKCNK3
SCHEMBL21588759 0.84 PTGS1 (0.72) PTGS1NPC1RAB9AKCNK3TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed
EP-0735403-B1 Liquid crystal orienting agent JSR CORP (JP) 2004-03-17 EP disclosed
US-5700860-A Liquid crystal orienting agent JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1997-12-23 US disclosed
EP-0735403-A1 Liquid crystal orienting agent JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1996-10-02 EP disclosed