SCHEMBL6560100

SCHEMBL6560100

O=C(O)CN1[CH]C(NC(=O)C(CS(=O)(=O)Cc2ccccc2)NC(=O)N2CCOCC2)C1=O

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSS P25774 13/20 0.53
CTSB P07858 6/20 0.41
CTSL P07711 6/20 0.41
CTSK P43235 2/20 0.40
CTSH P09668 1/20 0.40
CTSC P53634 1/20 0.40
TACR2 P21452 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6848353 0.83 CTSS (0.54) CTSSCTSBCTSLCTSKCTSH
SCHEMBL6848124 0.82 CTSS (0.55) CTSSCTSBCTSLCTSKCTSH
SCHEMBL6848372 0.80 CTSS (0.52) CTSSCTSBCTSLCTSK
SCHEMBL14491119 0.80 CTSS (0.52) CTSSCTSBCTSLCTSK
SCHEMBL5438934 0.80 CTSS (0.57) CTSSCTSBCTSLCTSKCTSH
SCHEMBL3023908 0.80 CTSS (0.57) CTSSCTSBCTSLCTSKCTSH
SCHEMBL3023913 0.80 CTSS (0.57) CTSSCTSBCTSLCTSKCTSH
SCHEMBL6848129 0.79 CTSS (0.53) CTSSCTSBCTSLCTSKCTSH
SCHEMBL6847753 0.77 CTSS (0.49) CTSSCTSBCTSLCTSKCTSH
SCHEMBL6847162 0.77 CTSS (0.49) CTSSCTSBCTSLCTSKCTSH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1436255-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS CATHEPSIN INHIBITORS Aventis Pharmaceuticals, Inc. (US) 2004-07-14 EP disclosed
WO-2003024924-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS CATHEPSIN INHIBITORS AVENTIS PHARMACEUTICALS INC. (US) 2003-03-27 WO disclosed