SCHEMBL6561208

SCHEMBL6561208

COCCC(=O)Nc1cccc([C]=O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.50
MAP4K4 O95819 1/20 0.48
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
LMNA P02545 1/20 0.47
HTT P42858 1/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP2D6 P10635 1/20 0.47
GAA P10253 1/20 0.47
ALOX15 P16050 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
THRB P10828 1/20 0.46
HDAC3 O15379 1/20 0.46
EGFR P00533 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4085439 0.84 NPC1 (0.57) RAB9AHTTALDH1A1MAPTMTNR1B
SCHEMBL8880595 0.81 KDM4E (0.60) RAB9ACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL14948852 0.81 HDAC3 (0.64) RAB9ACYP1A2CYP3A4CYP2C19MEN1
SCHEMBL2702562 0.80 RAB9A (0.63) RAB9ACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL3217401 0.79 GAA (0.65) MEN1KMT2ALMNAALDH1A1GAA
SCHEMBL7452128 0.79 LMNA (0.57) RAB9AMEN1KMT2ALMNAALDH1A1
SCHEMBL10780717 0.79 LMNA (0.57) RAB9AMEN1KMT2ALMNAALDH1A1
SCHEMBL14405815 0.78 MAPT (0.68) RAB9AMAP4K4KMT2ALMNAHTT
SCHEMBL2971345 0.78 MAPT (0.52) RAB9AMAP4K4KMT2ALMNAHTT
SCHEMBL3469024 0.78 CYP3A4 (0.67) RAB9ACYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144365-B1 INHIBITORS OF ALPHA-4 BETA-1 MEDIATED CELL ADHESION TANABE SEIYAKU CO (JP) 2004-03-17 EP disclosed
EP-1144365-A3 INHIBITORS OF ALPHA-4 BETA-1 MEDIATED CELL ADHESION TANABE SEIYAKU CO., LTD. (JP) 2003-07-09 EP disclosed
EP-1144365-A2 INHIBITORS OF ALPHA-4 BETA-1 MEDIATED CELL ADHESION TANABE SEIYAKU CO., LTD. (JP) 2001-10-17 EP disclosed
WO-2000037429-A2 INHIBITORS OF α4β1 MEDIATED CELL ADHESION TANABE SEIYAKU CO., LTD. (JP) 2000-06-29 WO disclosed