SCHEMBL6561562

SCHEMBL6561562

C=CCc1c(O)ccc2c1ccn2CC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 1/20 0.37
SRD5A1 P18405 1/20 0.36
MTNR1A P48039 1/20 0.35
XDH P47989 1/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
MAPT P10636 2/20 0.33
GABRA1 P14867 2/20 0.33
GABRB2 P47870 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 2/20 0.33
HTR2C P28335 1/20 0.33
ALDH2 P05091 1/20 0.33
GAA P10253 1/20 0.33
AKR1B1 P15121 1/20 0.33
HPGD P15428 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
PPARG P37231 1/20 0.33
PPARD Q03181 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002745 0.84 SRD5A1 (0.34) PLA2G2ASRD5A1XDHMEN1KMT2A
SCHEMBL6560541 0.80 HTR2C (0.36) ALDH1A1KDM4EHTR2CHPGDCNR1
SCHEMBL6561182 0.78 ALDH1A1 (0.47) PLA2G2AXDHMEN1KMT2AALDH1A1
SCHEMBL23397300 0.72 HTR2C (0.37) HTR2CCYP19A1
SCHEMBL6398012 0.72 SRD5A1 (0.49) SRD5A1MTNR1AXDHMEN1KMT2A
SCHEMBL6561697 0.71 BIRC5 (0.38) PLA2G2ASRD5A1XDHMEN1KMT2A
SCHEMBL7856928 0.71 SRD5A1 (0.40) PLA2G2ASRD5A1MEN1KMT2AMAPT
SCHEMBL323547 0.70 XDH (0.54) SRD5A1MTNR1AXDHMEN1KMT2A
SCHEMBL15835664 0.69 SRD5A1 (0.41) PLA2G2ASRD5A1MTNR1AXDHMEN1
SCHEMBL28274016 0.69 SRD5A1 (0.46) PLA2G2ASRD5A1MTNR1AXDHMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904079-B1 ANTIDIABETIC AGENTS MERCK & CO INC (US) 2004-03-24 EP disclosed
EP-0904079-A4 1999-05-06 EP disclosed
EP-0904079-A1 ANTIDIABETIC AGENTS Merck & Co., Inc. (US) 1999-03-31 EP disclosed
US-5859051-A ACETYLPHENOL DERIVATIVES MERCK & CO., INC. (US) 1999-01-12 US disclosed
WO-1997027857-A1 ANTIDIABETIC AGENTS MERCK & CO., INC. (US) 1997-08-07 WO disclosed