SCHEMBL6561874

SCHEMBL6561874

CNC(=O)/C=C(\c1ccc(C(F)(F)F)cc1)c1cccc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.47
CNR2 P34972 3/20 0.43
KCNJ11 Q14654 1/20 0.43
RXFP1 Q9HBX9 2/20 0.41
DRD4 P21917 1/20 0.41
NPC1 O15118 1/20 0.41
CRHBP P24387 1/20 0.41
RAB9A P51151 1/20 0.41
CRHR2 Q13324 1/20 0.41
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NR4A1 P22736 2/20 0.39
NR4A2 P43354 2/20 0.39
NR4A3 Q92570 2/20 0.39
HDAC8 Q9BY41 2/20 0.38
MMP3 P08254 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6562127 1.00 PLK1 (0.47) PLK1CNR2KCNJ11RXFP1DRD4
SCHEMBL6561900 0.81 NPC1 (0.51) PLK1CNR2NPC1RAB9AALDH1A1
SCHEMBL6560669 0.81 NPC1 (0.51) PLK1CNR2NPC1RAB9AALDH1A1
SCHEMBL6561880 0.79 PLK1 (0.48) PLK1CNR2KCNJ11NPC1RAB9A
SCHEMBL6560724 0.79 PLK1 (0.48) PLK1CNR2KCNJ11NPC1RAB9A
SCHEMBL6560727 0.79 PLK1 (0.48) PLK1CNR2KCNJ11NPC1RAB9A
SCHEMBL6561798 0.78 PLK1 (0.55) PLK1KCNJ11NPC1RAB9AALDH1A1
SCHEMBL6561799 0.78 PLK1 (0.55) PLK1KCNJ11NPC1RAB9AALDH1A1
SCHEMBL6561794 0.78 PLK1 (0.55) PLK1KCNJ11NPC1RAB9AALDH1A1
SCHEMBL6563174 0.76 PLK1 (0.53) PLK1RXFP1NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944581-A4 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES LILLY CO ELI (US) 2004-09-08 EP disclosed
EP-0944581-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1999-09-29 EP disclosed
WO-1998022429-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1998-05-28 WO disclosed