SCHEMBL6560669

SCHEMBL6560669

CNC(=O)/C=C(/c1ccc(OC)cc1)c1cccc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.51
KMT2A Q03164 3/20 0.51
RAB9A P51151 2/20 0.51
GCGR P47871 1/20 0.51
MTNR1A P48039 1/20 0.49
PLK1 P53350 2/20 0.48
CACNA1B Q00975 1/20 0.46
APBA1 Q02410 1/20 0.46
ALDH1A1 P00352 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
POLB P06746 1/20 0.46
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44
LMNA P02545 1/20 0.44
CNR2 P34972 3/20 0.44
CNR1 P21554 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6561900 1.00 NPC1 (0.51) NPC1KMT2ARAB9AGCGRMTNR1A
SCHEMBL1176798 0.86 NPC1 (0.51) NPC1KMT2ARAB9AGCGRCACNA1B
SCHEMBL6561769 0.85 NPC1 (0.43) NPC1KMT2ARAB9AGCGRMTNR1A
SCHEMBL6561831 0.85 NPC1 (0.43) NPC1KMT2ARAB9AGCGRMTNR1A
SCHEMBL6560697 0.83 NPC1 (0.51) NPC1KMT2ARAB9APLK1ALDH1A1
SCHEMBL6561877 0.83 NPC1 (0.51) NPC1KMT2ARAB9APLK1ALDH1A1
SCHEMBL6562127 0.81 PLK1 (0.47) NPC1RAB9APLK1ALDH1A1SMN1; SMN2
SCHEMBL6561874 0.81 PLK1 (0.47) NPC1RAB9APLK1ALDH1A1SMN1; SMN2
SCHEMBL6560672 0.80 CACNA1B (0.52) NPC1KMT2ARAB9AGCGRMTNR1A
SCHEMBL9856912 0.80 GCGR (0.67) NPC1KMT2ARAB9AGCGRMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944581-A4 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES LILLY CO ELI (US) 2004-09-08 EP disclosed
EP-0944581-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1999-09-29 EP disclosed
WO-1998022429-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1998-05-28 WO disclosed