SCHEMBL6562196

SCHEMBL6562196

Oc1ccccc1-n1ccc(-c2ccccc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.50
KDM4E B2RXH2 3/20 0.48
MAPT P10636 1/20 0.48
XBP1 P17861 1/20 0.48
MAPK1 P28482 1/20 0.48
COMT P21964 4/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC4 P56524 1/20 0.41
HDAC2 Q92769 1/20 0.41
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40
TUBB2A Q13885 1/20 0.40
TUBB8 Q3ZCM7 1/20 0.40
TUBA3E Q6PEY2 1/20 0.40
TUBA1A Q71U36 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28059853 0.77 BCHE (0.49) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL18612923 0.74 IDO1 (0.55) IDO1KDM4EMAPTXBP1MAPK1
SCHEMBL2589320 0.74 IDO1 (0.47) IDO1KDM4EMAPTXBP1MAPK1
SCHEMBL28329739 0.74 MGLL (0.46) MAPTALDH1A1HPGDLMNAIDH1
SCHEMBL12332875 0.73 IDH1 (0.53) KDM4EMAPTXBP1MAPK1COMT
SCHEMBL6559666 0.73 TUBB4A (0.49) KDM4EMAPTTUBB4ATUBBTUBA3C
SCHEMBL2050250 0.72 IDO1 (0.57) IDO1KDM4EMAPTXBP1MAPK1
SCHEMBL4719825 0.70 IDO1 (0.43) IDO1KDM4EMAPTXBP1MAPK1
SCHEMBL28667917 0.69 IDO1 (0.50) IDO1KDM4EMAPTXBP1MAPK1
SCHEMBL1535129 0.69 IDO1 (0.59) IDO1KDM4EMAPTXBP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1071670-B1 NOVEL DIPHENYL-SUBSTITUTED 5-RING-HETEROCYCLES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA (DE) 2004-07-07 EP disclosed
US-6255327-B1 ANTIHYPOXC, ANTIISCHEMIC AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-07-03 US disclosed
EP-1071670-A1 NOVEL DIPHENYL-SUBSTITUTED 5-RING-HETEROCYCLES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-01-31 EP disclosed
WO-1999054314-A1 NOVEL DIPHENYL-SUBSTITUTED 5-RING-HETEROCYCLES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-28 WO disclosed