SCHEMBL6562369

SCHEMBL6562369

CC(O)(C(=O)N(c1ccccc1)S(=O)(=O)c1ccccc1)C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.54
ABCC9 O60706 2/20 0.53
ABCC8 Q09428 2/20 0.53
KCNJ11 Q14654 2/20 0.53
KCNJ8 Q15842 2/20 0.53
NR1H3 Q13133 6/20 0.50
HSD11B1 P28845 2/20 0.48
NR1H2 P55055 6/20 0.48
MEN1 O00255 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
NR1I2 O75469 3/20 0.46
RORC P51449 2/20 0.45
RORA P35398 1/20 0.45
RORB Q92753 1/20 0.45
NR1H4 Q96RI1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7247986 0.84 ABCC9 (0.45) KMT2AABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8657172 0.84 ABCC9 (0.45) KMT2AABCC9ABCC8KCNJ11KCNJ8
SCHEMBL31211576 0.83 KMT2A (0.57) KMT2ANR1H3NR1H2MEN1NR1I2
SCHEMBL8657904 0.82 ABCC9 (0.47) KMT2AABCC9ABCC8KCNJ11KCNJ8
Dimethylamine SCHEMBL6569138 0.79 ABCC9 (0.44) KMT2AABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8656072 0.79 ABCC9 (0.44) KMT2AABCC9ABCC8KCNJ11KCNJ8
SCHEMBL6569133 0.78 ABCC9 (0.44) KMT2AABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7253590 0.78 ABCC9 (0.41) KMT2AABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7247433 0.78 ABCC9 (0.44) KMT2AABCC9ABCC8KCNJ11KCNJ8
Dimethylamine SCHEMBL6571779 0.77 ABCC9 (0.43) KMT2AABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214296-B1 SUBSTITUTED N-PHENYL 2-HYDROXY-2-METHYL-3,3,3-TRIFLUOROPROPANAMIDE DERIVATIVES WHICH ELEVATE PYRUVATE DEHYDROGENASE ACTIVITY ASTRAZENECA AB (SE) 2004-03-24 EP disclosed