SCHEMBL6562453

SCHEMBL6562453

COC(=O)C1=C(C)C(=O)CCC1(C)C

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.38
MAPT P10636 1/20 0.37
ALOX15 P16050 1/20 0.37
SRD5A1 P18405 2/20 0.35
SRD5A2 P31213 2/20 0.35
ALDH1A1 P00352 2/20 0.35
TSHR P16473 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
GAA P10253 1/20 0.33
KDM4E B2RXH2 2/20 0.32
CASP1 P29466 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PKM P14618 1/20 0.32
HPGD P15428 2/20 0.32
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7708414 0.83 MAPT (0.43) TRPA1MAPTALOX15
SCHEMBL10650334 0.83 KDM4E (0.42) TRPA1MAPTALOX15SRD5A1SRD5A2
SCHEMBL11812280 0.81 ALDH1A1 (0.40) MAPTSRD5A1SRD5A2ALDH1A1TSHR
SCHEMBL11394565 0.79 MAPT (0.40) TRPA1MAPTALOX15
SCHEMBL6562444 0.76 CYP1A2 (0.32)
SCHEMBL10457193 0.74 MAPT (0.39) TRPA1MAPTALOX15
SCHEMBL12160497 0.73 CYP1A2 (0.44) TRPA1MAPTALOX15ALDH1A1TSHR
SCHEMBL7171679 0.73 CYP1A2 (0.44) TRPA1MAPTALOX15ALDH1A1TSHR
SCHEMBL22077241 0.73 SLC6A3 (0.34) TSHRSMN1; SMN2
SCHEMBL10380096 0.72 MAPT (0.41) TRPA1MAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017180248-A9 ENANTIOENRICHED VIRIDICATUMTOXIN B ANALOGS WILLIAM MARSH RICE UNIVERSITY (US) 2018-11-01 WO disclosed
WO-2017180248-A1 ENANTIOENRICHED VIRIDICATUMTOXIN B ANALOGS WILLIAM MARSH RICE UNIVERSITY (US) 2017-10-19 WO disclosed
WO-2017180248-A1 ENANTIOENRICHED VIRIDICATUMTOXIN B ANALOGS WILLIAM MARSH RICE UNIVERSITY (US) 2017-10-19 WO disclosed
EP-1144365-B1 INHIBITORS OF ALPHA-4 BETA-1 MEDIATED CELL ADHESION TANABE SEIYAKU CO (JP) 2004-03-17 EP disclosed