SCHEMBL6563293

SCHEMBL6563293

Cc1cc(C#CCNc2ccc(C#N)cc2)ccc1C(=O)n1ccnc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.43
LRRK2 Q5S007 2/20 0.36
CD38 P28907 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CACNA1B Q00975 1/20 0.35
ACACB O00763 1/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
GRK2 P25098 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
GRM5 P41594 2/20 0.34
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565363 0.78 GAA (0.41) LRRK2ALDH1A1L3MBTL1
SCHEMBL6562060 0.76 PLA2G7 (0.39) LRRK2ALDH1A1GRM5NOS3NOS1
SCHEMBL6563213 0.75 KMT2A (0.39) LRRK2CYP11B1CYP11B2GRM5
SCHEMBL7808322 0.75 NPC1 (0.39) LRRK2GRK2GRM5NOS3NOS1
SCHEMBL6563806 0.74 ACACB (0.52) ACACB
SCHEMBL4810734 0.72 CYP19A1 (0.68) CYP19A1CD38ALDH1A1CYP11B1CYP11B2
SCHEMBL17039626 0.71 CYP19A1 (0.52) CYP19A1CD38ALDH1A1CACNA1BCYP11B1
SCHEMBL5885749 0.71 ACACB (0.48) ALDH1A1ACACB
SCHEMBL5885707 0.71 ACACB (0.38) ALDH1A1ACACBGRM5
SCHEMBL18184936 0.70 CYP19A1 (0.56) CYP19A1CD38ALDH1A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed