SCHEMBL6563708

SCHEMBL6563708

CCOC(=O)CCN(C(=O)c1ccc(CC)c(C#CCNc2ccc(C(=N)NC(=O)OC(C)(C)C)cc2)c1)c1ccccn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
F2 P00734 6/20 0.41
NR1I2 O75469 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
SLC6A2 P23975 1/20 0.41
AGTR1 P30556 1/20 0.41
SLC6A3 Q01959 1/20 0.41
SCN5A Q14524 1/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPK1 P28482 2/20 0.41
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SLC22A2 O15244 1/20 0.39
F10 P00742 1/20 0.39
PLG P00747 1/20 0.39
PLAT P00750 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6564395 0.88 NQO2 (0.63) NQO2SMN1; SMN2HSD17B10F2NR1I2
SCHEMBL6565269 0.84 ALDH1A1 (0.45) NQO2SMN1; SMN2HSD17B10F2NR1I2
SCHEMBL6565428 0.82 MEN1 (0.34) NQO2SMN1; SMN2HSD17B10F2ALDH1A1
SCHEMBL6565360 0.79 F2 (0.59) NQO2SMN1; SMN2HSD17B10F2SLC22A2
SCHEMBL6563093 0.77 NQO2 (0.32) NQO2F2ALDH1A1MAPK1MEN1
SCHEMBL6563344 0.75 NQO2 (0.33) NQO2
SCHEMBL6563537 0.74 PLAU (0.38) KMT2A
SCHEMBL6565418 0.74 MEN1 (0.33) SMN1; SMN2HSD17B10F2ALDH1A1MAPK1
SCHEMBL6561955 0.73 SMN1; SMN2 (0.31) SMN1; SMN2MAPT
SCHEMBL6565414 0.73 PTPN11 (0.33) NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed