SCHEMBL6564992

SCHEMBL6564992

N#CC1CCCC(N(C(=O)C2(OC(=O)Nc3ccc4ccccc4c3)CCCCC2)C2CCNC2)C1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 16/20 0.44
SLC6A2 P23975 15/20 0.44
SLC6A3 Q01959 6/20 0.44
KCNH2 Q12809 4/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
CYP2D6 P10635 1/20 0.35
EPHX1 P07099 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7431178 0.81 JAK3 (0.38) SLC6A4SLC6A2SLC6A3KCNH2USP2
SCHEMBL7436060 0.79 SLC6A4 (0.41) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL6564990 0.76 EPHX1 (0.36) SLC6A4SLC6A2SLC6A3USP2ALDH1A1
SCHEMBL6563732 0.73 ALDH1A1 (0.39) USP2ALDH1A1HPGDEPHX1MEN1
SCHEMBL6567334 0.70 SLC6A2 (0.44) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL3902181 0.63 CA12 (0.41) USP2ALDH1A1HPGDMEN1NPC1
SCHEMBL3907701 0.63 CTSS (0.41) USP2ALDH1A1HPGDEPHX1MEN1
SCHEMBL3907563 0.62 EPHX1 (0.41) USP2ALDH1A1HPGDCYP2D6EPHX1
SCHEMBL3909371 0.61 ALDH1A1 (0.41) USP2ALDH1A1HPGDCYP2D6EPHX1
SCHEMBL3894089 0.61 CA12 (0.45) USP2ALDH1A1HPGDCYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed