SCHEMBL6566917

SCHEMBL6566917

Cc1c(Cl)cc(NCc2ccc(Br)s2)c(O)c1Cl

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.33
POLB P06746 1/20 0.32
KDM4C Q9H3R0 1/20 0.31
HDAC1 Q13547 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4345532 0.81 EGFR (0.34) EGFRPOLB
SCHEMBL4354194 0.80 KMT2A (0.39) EGFRPOLB
SCHEMBL4352970 0.75 EGFR (0.38) EGFRPOLBHDAC8
SCHEMBL4353715 0.75 EGFR (0.41) EGFRHDAC1HDAC6
SCHEMBL4351839 0.73 HDAC8 (0.45) HDAC1HDAC8HDAC6
SCHEMBL6568648 0.73 LMNA (0.41)
SCHEMBL6566390 0.72 BRD4 (0.48) POLBKDM4C
SCHEMBL4347039 0.72 APP (0.48) POLB
SCHEMBL4345563 0.70 BRD4 (0.49)
SCHEMBL4358645 0.70 EGFR (0.45) EGFRKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed