SCHEMBL6567675

SCHEMBL6567675

O=C(CC12CC3CC(CC(C3)C1)C2)Nc1cc(Cl)c(O)c(Cl)c1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 7/20 0.65
P2RX5 Q93086 1/20 0.56
P2RX4 Q99571 1/20 0.56
P2RX2 Q9UBL9 1/20 0.56
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
GPR55 Q9Y2T6 1/20 0.52
USP2 O75604 1/20 0.52
CA12 O43570 1/20 0.52
CA9 Q16790 1/20 0.52
EPHX2 P34913 1/20 0.50
POLB P06746 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3321984 0.84 P2RX7 (0.72) P2RX7MEN1KMT2AGPR55USP2
SCHEMBL6941695 0.83 P2RX7 (0.65) P2RX7MEN1KMT2AGPR55USP2
SCHEMBL6939890 0.81 P2RX7 (0.70) P2RX7MEN1KMT2AGPR55USP2
SCHEMBL6940565 0.78 P2RX7 (1.00) P2RX7MEN1KMT2AUSP2
SCHEMBL6941699 0.78 P2RX7 (0.70) P2RX7MEN1KMT2AGPR55USP2
SCHEMBL12932448 0.77 P2RX7 (0.75) P2RX7MEN1KMT2AGPR55USP2
SCHEMBL4348906 0.77 EPHX2 (0.73) P2RX7P2RX5P2RX4P2RX2MEN1
SCHEMBL6941160 0.75 P2RX7 (0.67) P2RX7KMT2AGPR55EPHX2POLB
SCHEMBL11884308 0.75 P2RX7 (1.00) P2RX7MEN1KMT2AGPR55USP2
SCHEMBL6941644 0.74 P2RX7 (1.00) P2RX7EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed