SCHEMBL6568226

SCHEMBL6568226

CN(C)C(=O)Oc1ccc(C[C@H](NC(=O)[C@H]2CCCC[C@@H]2Cc2cc(F)cc(F)c2)C(=O)O)cc1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 19/20 0.44
ITGA4 P13612 18/20 0.44
ITGB3 P05106 1/20 0.41
ITGAV P06756 1/20 0.41
ITGA5 P08648 1/20 0.41
ITGB7 P26010 1/20 0.38
BCHE P06276 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7229806 0.90 ITGB1 (0.44) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL7225170 0.90 ITGB1 (0.44) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL6568926 0.90 ITGB1 (0.44) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL6568912 0.89 ITGB1 (0.51) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL6568334 0.87 ITGB1 (0.49) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL6569673 0.84 ITGB1 (0.52) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL5679763 0.72 ITGB1 (0.55) ITGB1ITGA4
SCHEMBL5859856 0.72 ITGA4 (0.46) ITGB1ITGA4ITGB7
SCHEMBL3855807 0.72 ITGB1 (0.56) ITGB1ITGA4ITGAVITGA5ITGB7
SCHEMBL4957436 0.72 ITGB1 (0.58) ITGB1ITGA4ITGAVITGA5ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161416-B1 ALPHA-AMINOACETIC ACID DERIVATIVES USEFUL AS ALPHA 4 BETA 7 - RECEPTOR ANTAGONISTS ELAN PHARM INC (US) 2004-04-14 EP claimed
US-6545160-B2 Alpha-aminoacetic acid derivatives bind alpha 4 beta 7 integrin, useful for treatment of inflammatory diseases in mammalian patient, such as asthma, Alzheimer's disease, atherosclerosis, AIDS dementia, diabetes, rheumatoid arthritis ELAN PHARMACEUTICALS, INC. 2003-04-08 US disclosed