SCHEMBL6568912

SCHEMBL6568912

CN(C)C(=O)Oc1ccc(C[C@H](NC(=O)[C@H]2CCCC[C@@H]2Cc2ccccc2)C(=O)O)cc1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 15/20 0.51
ITGA4 P13612 14/20 0.51
ITGB3 P05106 1/20 0.45
ITGAV P06756 1/20 0.45
ITGA5 P08648 1/20 0.45
LMNA P02545 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ITGB7 P26010 1/20 0.44
ALDH1A1 P00352 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6568334 0.92 ITGB1 (0.49) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL6569673 0.90 ITGB1 (0.52) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL6568226 0.89 ITGB1 (0.44) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL7225170 0.88 ITGB1 (0.44) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL6568926 0.88 ITGB1 (0.44) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL7229806 0.88 ITGB1 (0.44) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL7224863 0.81 ITGB1 (0.47) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL7230074 0.81 ITGB1 (0.48) ITGB1ITGA4ITGB3ITGAVITGA5
SCHEMBL5679669 0.76 ITGB1 (0.63) ITGB1ITGA4ALDH1A1
SCHEMBL6568332 0.75 ITGA4 (0.47) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161416-B1 ALPHA-AMINOACETIC ACID DERIVATIVES USEFUL AS ALPHA 4 BETA 7 - RECEPTOR ANTAGONISTS ELAN PHARM INC (US) 2004-04-14 EP claimed
US-6545160-B2 Alpha-aminoacetic acid derivatives bind alpha 4 beta 7 integrin, useful for treatment of inflammatory diseases in mammalian patient, such as asthma, Alzheimer's disease, atherosclerosis, AIDS dementia, diabetes, rheumatoid arthritis ELAN PHARMACEUTICALS, INC. 2003-04-08 US disclosed