SCHEMBL6569987

SCHEMBL6569987

Cc1c(Sc2ccccc2)ccc([N+](=O)[O-])c1N

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.55
PDE7A Q13946 7/20 0.52
PDE7B Q9NP56 2/20 0.52
GSTP1 P09211 1/20 0.52
GSTM2 P28161 1/20 0.52
GAA P10253 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.48
HTT P42858 2/20 0.48
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
TDP1 Q9NUW8 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
POLB P06746 1/20 0.45
USP47 Q96K76 1/20 0.44
IDO1 P14902 1/20 0.44
ABCC9 O60706 1/20 0.44
ABCC8 Q09428 1/20 0.44
KCNJ11 Q14654 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11070941 0.82 PDE7A (0.60) MAPTPDE7APDE7BGSTP1GSTM2
SCHEMBL810289 0.75 PDE7A (0.68) MAPTPDE7APDE7BGSTP1GSTM2
SCHEMBL2968510 0.75 PDE7A (0.68) MAPTPDE7APDE7BGSTP1GSTM2
SCHEMBL11495179 0.75 PDE7A (0.51) MAPTPDE7APDE7BGSTP1GSTM2
SCHEMBL30338244 0.73 PDE7A (0.65) MAPTPDE7APDE7BGSTP1GSTM2
SCHEMBL1713219 0.73 PDE7A (0.65) MAPTPDE7APDE7BGSTP1GSTM2
Acetic Acid SCHEMBL8213274 0.73 MAPT (0.67) MAPTPDE7APDE7BGSTP1GSTM2
SCHEMBL15155301 0.73 PDE7A (0.60) MAPTPDE7APDE7BGSTP1GSTM2
SCHEMBL4707544 0.72 PDE7A (0.48) MAPTPDE7APDE7BGSTP1GSTM2
SCHEMBL9808890 0.72 PDE7A (0.49) MAPTPDE7APDE7BGSTP1GSTM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091935-B1 METHOD FOR PREPARING 2-NITRO-5-(PHENYLTHIO)-ANILINES BAYER CHEMICALS AG (DE) 2004-04-21 EP disclosed
US-6552230-B1 Amination of a 2,4-dichloronitrobenzene with ammonia forming 5-chloro-2-nitroaniline which is reacted with a thiophenol; one pot process BAYER AKTIENGESELLSCHAFT (DE) 2003-04-22 US disclosed
EP-1091935-A2 METHOD FOR PREPARING 2-NITRO-5-(PHENYLTHIO)-ANILINES Bayer Aktiengesellschaft (DE) 2001-04-18 EP disclosed
WO-2000001669-A2 METHOD FOR PREPARING 2-NITRO-5-(PHENYLTHIO)-ANILINES BAYER AKTIENGESELLSCHAFT (DE) 2000-01-13 WO disclosed
EP-0061110-B1 NITRO-ANILINES CELAMERCK GmbH & Co. KG (DE) 1984-08-08 EP disclosed
EP-0061110-A1 Nitro-anilines CELAMERCK GmbH & Co. KG (DE) 1982-09-29 EP disclosed