SCHEMBL6570672

SCHEMBL6570672

Nc1ccc(N)c(-c2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.58
MAPK1 P28482 1/20 0.58
RORC P51449 2/20 0.54
RORB Q92753 2/20 0.54
ADORA2A P29274 2/20 0.48
ADORA1 P30542 2/20 0.48
MAOB P27338 4/20 0.46
KDM1A O60341 2/20 0.45
ABCG2 Q9UNQ0 1/20 0.44
IKBKB O14920 1/20 0.43
BRD4 O60885 1/20 0.43
HRH1 P35367 1/20 0.42
HRH4 Q9H3N8 1/20 0.42
XDH P47989 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
KIF11 P52732 2/20 0.41
IDO1 P14902 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6572095 0.98 TSHR (0.56) TSHRMAPK1RORCRORBADORA2A
SCHEMBL5851547 0.88 TSHR (0.60) TSHRMAPK1RORCRORBADORA2A
SCHEMBL6011230 0.86 TSHR (0.58) TSHRMAPK1RORCRORBADORA2A
SCHEMBL3786041 0.86 TSHR (0.58) TSHRMAPK1RORCRORBADORA2A
SCHEMBL28676842 0.83 TSHR (0.55) TSHRMAPK1RORCRORBADORA2A
SCHEMBL21019702 0.83 RORB (0.62) TSHRMAPK1RORCRORBADORA2A
SCHEMBL398678 0.82 ADORA2A (0.54) TSHRMAPK1RORCRORBADORA2A
SCHEMBL2573330 0.81 TSHR (0.56) TSHRMAPK1RORCRORBADORA2A
SCHEMBL5687763 0.81 RORB (0.56) TSHRMAPK1RORCRORBADORA2A
SCHEMBL22345011 0.81 MAOA (0.44) TSHRMAPK1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed