SCHEMBL6571132

SCHEMBL6571132

Nc1ccc(NCC(O)CO)c(-c2cccc([N+](=O)[O-])c2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
GLA P06280 1/20 0.41
MAPT P10636 3/20 0.41
GAA P10253 2/20 0.41
KDM4E B2RXH2 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HDAC2 Q92769 1/20 0.39
PKM P14618 2/20 0.39
PTPRC P08575 1/20 0.39
MAPK1 P28482 1/20 0.39
MITF O75030 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ADRB2 P07550 2/20 0.38
ADRB1 P08588 2/20 0.38
ADRB3 P13945 2/20 0.38
AKR1C3 P42330 2/20 0.37
AKR1C2 P52895 2/20 0.37
CA1 P00915 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6571859 0.86 KDM4E (0.37) ALDH1A1MAPTKDM4E
SCHEMBL6571992 0.84 PKM (0.52) ALDH1A1MAPTGAAKDM4EL3MBTL1
SCHEMBL6572033 0.83 MYC (0.48) ALDH1A1GLAMAPTGAAMEN1
SCHEMBL6571461 0.82 CHEK1 (0.41)
SCHEMBL6572232 0.81 PIK3CG (0.38) ALDH1A1CA1CA2
Hydrochloric Acid SCHEMBL6572537 0.81 CHEK1 (0.40)
SCHEMBL6572450 0.80 ADORA1 (0.37) ALDH1A1
SCHEMBL6571398 0.80 TAAR1 (0.41) MAPK1
SCHEMBL6571424 0.80 EGFR (0.39) MAPTKDM4EMEN1KMT2A
SCHEMBL6572773 0.80 MAPT (0.41) ALDH1A1GLAMAPTGAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed