SCHEMBL6571244

SCHEMBL6571244

CC(=O)O[C@](C)(C(=O)Nc1ccc(Sc2ccc(NC(=O)Nc3ccccc3)cc2)cc1Cl)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 11/20 0.41
PDK2 Q15119 11/20 0.41
PDK3 Q15120 11/20 0.41
PDK4 Q16654 11/20 0.41
NR1H2 P55055 2/20 0.39
NR1H3 Q13133 2/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
NPC1 O15118 2/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
CA12 O43570 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6571253 1.00 PDK1 (0.41) PDK1PDK2PDK3PDK4NR1H2
SCHEMBL6568763 0.90 HTT (0.42) PDK1PDK2PDK3PDK4MEN1
SCHEMBL6568770 0.90 HTT (0.42) PDK1PDK2PDK3PDK4MEN1
SCHEMBL6348658 0.88 PDK1 (0.41) PDK1PDK2PDK3PDK4MEN1
SCHEMBL6348654 0.88 PDK1 (0.41) PDK1PDK2PDK3PDK4MEN1
SCHEMBL6358529 0.86 ALDH1A1 (0.48) PDK1PDK2PDK3PDK4MEN1
SCHEMBL6358525 0.86 ALDH1A1 (0.48) PDK1PDK2PDK3PDK4MEN1
SCHEMBL6351405 0.86 PDK1 (0.44) PDK1PDK2PDK3PDK4CA1
SCHEMBL6351400 0.86 PDK1 (0.44) PDK1PDK2PDK3PDK4CA1
SCHEMBL6568932 0.85 PDK1 (0.58) PDK1PDK2PDK3PDK4NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082110-B1 USE OF COMPOUNDS FOR THE ELEVATION OF PYRUVATE DEHYDROGENASE ACTIVITY ASTRAZENECA AB (SE) 2004-03-24 EP disclosed