SCHEMBL6571640

SCHEMBL6571640

CCCCCCCC(=O)N[C@H](c1ccccc1)[C@@H](O)CO

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CERT1 Q9Y5P4 3/20 0.65
ASAH1 Q13510 2/20 0.64
ALDH1A1 P00352 1/20 0.64
ACER2 Q5QJU3 1/20 0.64
UGCG Q16739 2/20 0.53
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
SMPD2 O60906 2/20 0.51
SMPD1 P17405 1/20 0.51
TP53 P04637 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
NFKB1 P19838 1/20 0.50
MAPK1 P28482 1/20 0.50
CYP2C19 P33261 1/20 0.50
HIF1A Q16665 1/20 0.50
MAPT P10636 1/20 0.50
MTOR P42345 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27357411 0.83 ASAH1 (0.63) CERT1ASAH1ALDH1A1ACER2UGCG
SCHEMBL8666377 0.83 ASAH1 (0.63) CERT1ASAH1ALDH1A1ACER2UGCG
SCHEMBL14960683 0.82 ASAH1 (0.61) CERT1ASAH1ALDH1A1ACER2UGCG
SCHEMBL6570067 0.82 ASAH1 (0.68) CERT1ASAH1ALDH1A1ACER2
SCHEMBL8338663 0.82 ASAH1 (0.68) CERT1ASAH1ALDH1A1ACER2
SCHEMBL7769012 0.82 ASAH1 (0.68) CERT1ASAH1ALDH1A1ACER2
SCHEMBL7769010 0.82 ASAH1 (0.68) CERT1ASAH1ALDH1A1ACER2
SCHEMBL8341808 0.81 ALDH1A1 (0.71) CERT1ASAH1ALDH1A1ACER2UGCG
SCHEMBL7773484 0.81 ALDH1A1 (0.71) CERT1ASAH1ALDH1A1ACER2UGCG
SCHEMBL7773486 0.81 ALDH1A1 (0.71) CERT1ASAH1ALDH1A1ACER2UGCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1156054-B1 DRUGS CONTAINING PHOSPHORIC ACID DERIVATIVES AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-04-14 EP disclosed
US-6495533-B1 TUMOR NECROSIS FACTOR INHIBITORS; RHEUMATOID ARTHRITIS, ULCERATIVE COLITIS, CROHN'S DISEASE, HEPATITIS, SEPSIS, HEMORRHAGIC SHOCK, MULTIPLE SCLEROSIS, CEREBRAL INFARCTION, DIABETES, INTERSTITIAL PNEUMONIA, PAIN, HIV ONO PHARMACEUTICAL CO., LTD. (JP) 2002-12-17 US disclosed
EP-1156054-A1 DRUGS CONTAINING PHOSPHORIC ACID DERIVATIVES AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-11-21 EP disclosed