SCHEMBL6571824

SCHEMBL6571824

Nc1ccc(NCC(O)CO)c(-c2ccc(Cl)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
AR P10275 2/20 0.34
VDR P11473 2/20 0.34
KIT P10721 1/20 0.33
PRKCA P17252 1/20 0.33
GSK3B P49841 1/20 0.33
PPARG P37231 1/20 0.33
BCHE P06276 1/20 0.33
F10 P00742 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6574847 0.91 PDE3B (0.37) CYP1A2PDE3BPDE3AARVDR
SCHEMBL6573407 0.87 USP7 (0.36) PDE3BPDE3AARVDR
SCHEMBL6572042 0.87 PDE3B (0.34) CYP1A2PDE3BPDE3AARVDR
SCHEMBL6572450 0.87 ADORA1 (0.37) PRKCAGSK3B
SCHEMBL6571431 0.86 AR (0.36) CYP1A2PDE3BPDE3AARVDR
SCHEMBL6573194 0.86 SCN9A (0.38) CYP1A2PDE3BPDE3APRKCAGSK3B
SCHEMBL6572423 0.86 PDE3B (0.34) CYP1A2PDE3BPDE3AARVDR
SCHEMBL6571878 0.86 CYP1A2 (0.38) CYP1A2PDE3BPDE3A
SCHEMBL6571461 0.86 CHEK1 (0.41)
SCHEMBL6571859 0.84 KDM4E (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed