SCHEMBL6572213

SCHEMBL6572213

CC(C)OC(=O)c1cccc(-c2ccc(C(=O)O)cc2)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.69
CD274 Q9NZQ7 1/20 0.69
RXRA P19793 4/20 0.64
RXRB P28702 4/20 0.64
RXRG P48443 1/20 0.59
BCL2 P10415 1/20 0.55
SMN1; SMN2 Q16637 4/20 0.54
NPC1 O15118 4/20 0.54
RAB9A P51151 4/20 0.54
MAPT P10636 2/20 0.54
HTT P42858 2/20 0.54
ALDH1A1 P00352 2/20 0.53
KMO O15229 1/20 0.53
LMNA P02545 2/20 0.52
GAA P10253 1/20 0.52
CA12 O43570 1/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA7 P43166 1/20 0.51
CA9 Q16790 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20085587 0.85 PDCD1 (0.59) PDCD1CD274RXRARXRBRXRG
SCHEMBL20085556 0.85 PDCD1 (0.59) PDCD1CD274RXRARXRBRXRG
SCHEMBL6233392 0.84 NPC1 (0.62) PDCD1CD274RXRARXRBSMN1; SMN2
SCHEMBL30678268 0.84 NPC1 (0.62) PDCD1CD274RXRARXRBSMN1; SMN2
SCHEMBL14524832 0.83 PDCD1 (0.57) PDCD1CD274RXRARXRBRXRG
SCHEMBL7224347 0.83 CA12 (0.64) RXRARXRBRXRGBCL2KMO
Benzoic Acid 1-Methylethyl Ester SCHEMBL28356777 0.82 PDCD1 (0.74) PDCD1CD274RXRARXRBSMN1; SMN2
SCHEMBL296543 0.82 PDCD1 (1.00) PDCD1CD274RXRARXRBSMN1; SMN2
Benzoic Acid 1-Methylethyl Ester SCHEMBL29187646 0.80 PDCD1 (0.70) PDCD1CD274SMN1; SMN2NPC1RAB9A
SCHEMBL69066 0.80 KMO (0.80) RXRARXRBRXRGBCL2KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140072-B1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-04-14 EP disclosed
EP-1140072-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2003-04-16 EP disclosed
EP-1140072-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2001-10-10 EP disclosed
WO-2000040239-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-13 WO disclosed