Bispyribac

Bispyribac

SCHEMBL65725

COc1cc(OC)nc(Oc2cccc(Oc3nc(OC)cc(OC)n3)c2C(=O)O)n1

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
CA7 P43166 1/20 0.56
CA9 Q16790 1/20 0.56
CA14 Q9ULX7 1/20 0.56
NPSR1 Q6W5P4 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
GAA P10253 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
ALDH1A1 P00352 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bispyribac SCHEMBL4895772 1.00 CA12 (0.56) CA12CA1CA2CA7CA9
Bispyribac SCHEMBL238471 0.98 CA12 (0.54) CA12CA1CA2CA7CA9
Bispyribac SCHEMBL9195440 0.98 CA12 (0.54) CA12CA1CA2CA7CA9
Bispyribac SCHEMBL2114791 0.98 CA12 (0.54) CA12CA1CA2CA7CA9
SCHEMBL8952122 0.97 CA12 (0.62) CA12CA1CA2CA7CA9
SCHEMBL9539769 0.96 LMNA (0.53) CA12CA1CA2CA7CA9
SCHEMBL13197224 0.93 CYP1A2 (0.51) CA12CA1CA2CA7CA9
SCHEMBL8801724 0.93 ALDH1A1 (0.63) NPSR1CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL9221672 0.93 CYP1A2 (0.57) NPSR1CYP1A2CYP3A4GAACYP2C9
Bispyribac SCHEMBL9197260 0.93 NPSR1 (0.51) NPSR1CYP1A2CYP3A4GAACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10248 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4713317-A1 A PROCESS FOR PURIFICATION OF ETHOFUMESATE Adama Agan Ltd. (IL) 2026-03-25 EP claimed
US-20260060254-A1 HERBICIDAL COMPOSITIONS BAYER AG (DE) 2026-03-05 US claimed
EP-4677099-A2 HERBICIDE-RESISTANT GENES FOR MITOCHONDRIAL TRANSFORMATION Napigen, Inc. (US) 2026-01-14 EP claimed
US-20260007133-A1 HERBICIDAL COMPOSITION COMPRISING AZINE COMPOUNDS BASF SE (DE) 2026-01-08 US claimed
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
US-20250318528-A1 HERBICIDE COMPOSITION AND WEED CONTROLLING METHOD SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2025-10-16 US claimed
EP-4601471-A1 SUBSTITUTED 5-MEMBERED RINGS AND THEIR USE AS PESTICIDES Corteva Agriscience LLC (US) 2025-08-20 EP claimed
EP-3578543-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-08-20 EP claimed
EP-4593598-A1 STORAGE-STABLE COMPOSITIONS INCLUDING BIXLOZONE AND BEFLUBUTAMID FMC Corporation (US) 2025-08-06 EP claimed
US-6207617-B1 POLYOXYETHYLENE GLYCOL C24-60 ALCOHOLATE SURFACTANT, HERBICIDES MONSANTO COMPANT 2001-03-27 US claimed
EP-1073331-A1 CONCENTRATE COMPOSITION OF PLANT TREATMENT COMPOUND IN ACID FORM MONSANTO COMPANY (US) 2001-02-07 EP claimed
WO-2000016627-A1 SYNERGISTIC ACTIVE SUBSTANCE COMBINATIONS FOR CONTROLLING HARMFUL PLANTS AVENTIS CROPSCIENCE GMBH (DE) 2000-03-30 WO claimed
WO-2000008932-A1 HERBICIDES WITH ACYLATED AMINOPHENYLSULFONYL UREA AVENTIS CROPSCIENCE GMBH (DE) 2000-02-24 WO claimed
WO-2000008937-A1 HERBICIDES FOR TOLERANT OR RESISTANT COTTON CULTURES AVENTIS CROPSCIENCE GMBH (DE) 2000-02-24 WO claimed
WO-2000003591-A2 HERBICIDES AVENTIS CROPSCIENCE GMBH (DE) 2000-01-27 WO claimed
WO-1999055155-A1 CONCENTRATE COMPOSITION OF PLANT TREATMENT COMPOUND IN ACID FORM MONSANTO COMPANY (US) 1999-11-04 WO claimed
EP-0321846-B1 Pyrimidine derivatives, processes for their production, and herbicidal method and compositions KUMIAI CHEMICAL INDUSTRY CO (JP) 1995-04-19 EP claimed
US-4906285-A Pyrimidine derivatives and herbicidal method and compositions KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1990-03-06 US claimed
EP-0321846-A2 Pyrimidine derivatives, processes for their production, and herbicidal method and compositions KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1989-06-28 EP claimed