SCHEMBL6572867

SCHEMBL6572867

COC(=O)[C@@H](N)Cc1ccc(NC(=O)S)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
PTPRB P23467 1/20 0.43
LTA4H P09960 2/20 0.43
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
ROCK2 O75116 1/20 0.40
PTGS2 P35354 1/20 0.40
SLC7A5 Q01650 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
CIT O14578 1/20 0.39
SAE1 Q9UBE0 1/20 0.39
UBA2 Q9UBT2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12028836 0.85 ALDH1A1 (0.46) ALDH1A1PTPRBLTA4HESR1ESR2
SCHEMBL15080944 0.85 ALDH1A1 (0.46) ALDH1A1PTPRBLTA4HESR1ESR2
SCHEMBL27278675 0.84 ALDH1A1 (0.45) ALDH1A1PTPRBLTA4HESR1ESR2
SCHEMBL20865324 0.84 CA12 (0.48) ALDH1A1CA12CA1CA2CA9
SCHEMBL11563068 0.84 ALDH1A1 (0.45) ALDH1A1PTPRBLTA4HESR1ESR2
SCHEMBL7902861 0.83 ALDH1A1 (0.49) ALDH1A1PTPRBLTA4HESR1ESR2
SCHEMBL27278672 0.82 L3MBTL1 (0.54) ALDH1A1PTPRBLTA4HCA12CA1
SCHEMBL22427551 0.82 L3MBTL1 (0.54) ALDH1A1PTPRBLTA4HCA12CA1
Hydrochloric Acid SCHEMBL7902859 0.81 ALDH1A1 (0.51) ALDH1A1PTPRBLTA4HESR1ESR2
SCHEMBL30519915 0.81 TP53 (0.54) ALDH1A1LTA4HCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1474405-A2 PROCESS FOR THE PREPARATION OF 4-HETERO-SUBSTITUTED PHENYLALANINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2004-11-10 EP disclosed
WO-2003068725-A2 PROCESS FOR THE PREPARATION OF 4-HETERO-SUBSTITUTED PHENYLALANINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2003-08-21 WO disclosed