SCHEMBL6573422

SCHEMBL6573422

Nc1ccc(N(CCO)CCO)cc1-c1cccc(Br)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.42
ADK P55263 2/20 0.36
MAPT P10636 4/20 0.35
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
RAB9A P51151 2/20 0.33
KDM4E B2RXH2 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HK1 P19367 1/20 0.33
HKDC1 Q2TB90 1/20 0.33
S100B P04271 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
GAA P10253 1/20 0.33
PKM P14618 1/20 0.33
HTT P42858 1/20 0.33
MCL1 Q07820 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6570998 0.86 MAPT (0.38) HRH3MAPTKMT2AMEN1ALDH1A1
SCHEMBL6573029 0.85 HRH3 (0.38) HRH3ADKMAPTKMT2AMEN1
SCHEMBL6571445 0.85 KMT2A (0.43) MAPTKMT2AMEN1ALDH1A1HPGD
SCHEMBL6571458 0.84 CYP3A4 (0.38) MAPTKMT2AMEN1ALDH1A1GAA
SCHEMBL6571005 0.84 TAAR1 (0.39) MAPTKMT2AMEN1RAB9AKDM4E
SCHEMBL6571939 0.83 STK4 (0.45) MAPTKMT2AMEN1RAB9ASMN1; SMN2
SCHEMBL6571701 0.83 MAPT (0.38) MAPTKMT2AMEN1ALDH1A1RAB9A
SCHEMBL6570969 0.83 ADK (0.36) ADKMAPTKMT2AMEN1ALDH1A1
SCHEMBL6570991 0.81 MEN1 (0.42) KMT2AMEN1HPGDRAB9AKDM4E
SCHEMBL6573465 0.80 KMO (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed