SCHEMBL6576807

SCHEMBL6576807

Cc1noc([C@H]2O[C@@H](n3cnc4c(N[C@H](C)Cc5ccccc5)ncnc43)[C@H](O)[C@@H]2O)n1

nearest known ligand 0.71

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.69
ADORA2B P29275 6/20 0.69
ADORA3 P0DMS8 2/20 0.69
TP53 P04637 1/20 0.69
CYP3A4 P08684 1/20 0.69
TSHR P16473 1/20 0.69
ALOX12 P18054 1/20 0.69
NFKB1 P19838 1/20 0.69
HIF1A Q16665 1/20 0.69
ALDH1A1 P00352 1/20 0.69
HPGD P15428 1/20 0.69
PMP22 Q01453 1/20 0.69
NPC1 O15118 1/20 0.69
ADORA1 P30542 1/20 0.69
RAB9A P51151 1/20 0.69
RXFP1 Q9HBX9 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10601257 0.83 ADORA2A (0.80) ADORA2AADORA2BADORA3TP53CYP3A4
SCHEMBL10601644 0.83 ADORA2A (0.80) ADORA2AADORA2BADORA3TP53CYP3A4
SCHEMBL10601251 0.83 ADORA2A (0.80) ADORA2AADORA2BADORA3TP53CYP3A4
SCHEMBL6576870 0.83 ADORA3 (0.52) ADORA2AADORA2BADORA3TSHRNFKB1
(S)-Pia SCHEMBL122932 0.82 ADORA2A (1.00) ADORA2AADORA2BADORA3TP53CYP3A4
(S)-Pia SCHEMBL6762494 0.82 ADORA2A (1.00) ADORA2AADORA2BADORA3TP53CYP3A4
(S)-Pia SCHEMBL29616978 0.82 ADORA2A (1.00) ADORA2AADORA2BADORA3TP53CYP3A4
(S)-Pia SCHEMBL14829806 0.82 ADORA2A (1.00) ADORA2AADORA2BADORA3TP53CYP3A4
(R)-Pia SCHEMBL8907369 0.82 ADORA2A (1.00) ADORA2AADORA2BADORA3TP53CYP3A4
(R)-Pia SCHEMBL29389146 0.82 ADORA2A (1.00) ADORA2AADORA2BADORA3TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1090019-B1 ADENOSINE DERIVATIVES GLAXO GROUP LTD (GB) 2004-09-29 EP disclosed
EP-1447407-A1 Adenosine derivatives GLAXO GROUP LIMITED (GB) 2004-08-18 EP disclosed