SCHEMBL6578591

SCHEMBL6578591

NNC(=O)c1ccc(C(F)(F)F)c(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
KDM4E B2RXH2 4/20 0.50
MAPT P10636 2/20 0.50
LMNA P02545 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
GAA P10253 1/20 0.46
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
RAB9A P51151 1/20 0.44
FOXO1 Q12778 1/20 0.43
MPO P05164 1/20 0.43
CYP3A4 P08684 1/20 0.43
KDM5A P29375 1/20 0.43
BLM P54132 1/20 0.43
GFER P55789 1/20 0.43
PMP22 Q01453 1/20 0.43
HIF1A Q16665 1/20 0.43
KCNQ3 O43525 1/20 0.43
KCNQ2 O43526 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3530983 0.87 KDR (0.53) ALDH1A1KDM4EMAPTLMNAL3MBTL1
SCHEMBL29620917 0.81 KCNQ3 (0.53) ALDH1A1KDM4EMAPTLMNAL3MBTL1
SCHEMBL17596247 0.81 KCNQ3 (0.53) ALDH1A1KDM4EMAPTLMNAL3MBTL1
SCHEMBL4294249 0.81 HSD11B1 (0.45) RAB9AHTTKDRMRGPRX4
Hydrochloric Acid SCHEMBL30536936 0.79 HSD11B1 (0.44) RAB9AHTTKDRMRGPRX4
SCHEMBL24400223 0.79 KMO (0.43) CYP1A2CYP2D6CYP2C19RAB9AFOXO1
SCHEMBL9526608 0.79 NOTUM (0.46) CYP1A2CYP2D6CYP2C19RAB9AFOXO1
SCHEMBL1920001 0.79 TSHR (0.59) ALDH1A1MAPTKDRMRGPRX4
SCHEMBL29624981 0.79 TSHR (0.59) ALDH1A1MAPTKDRMRGPRX4
SCHEMBL30255650 0.79 NOTUM (0.46) CYP1A2CYP2D6CYP2C19RAB9AFOXO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1148357-C Triazole and imidazole derivative - 2004-05-05 CN disclosed
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
CN-1281852-A Triazole and imidazole derivative HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed