SCHEMBL6578700

SCHEMBL6578700

CCOc1ccc(C(=O)NN)cc1F

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 1/20 0.60
KCNQ2 O43526 1/20 0.60
TAS1R3 Q7RTX0 2/20 0.50
TAS1R1 Q7RTX1 2/20 0.50
RAB9A P51151 2/20 0.50
NPC1 O15118 1/20 0.50
USP2 O75604 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
HSD17B10 Q99714 1/20 0.50
CREBBP Q92793 1/20 0.49
HDAC1 Q13547 2/20 0.48
HDAC3 O15379 1/20 0.48
HDAC2 Q92769 1/20 0.48
TP53 P04637 1/20 0.48
MAPK1 P28482 3/20 0.48
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
KDM1A O60341 2/20 0.46
TSHR P16473 1/20 0.45
LMNA P02545 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6580973 0.86 KCNQ3 (0.45) KCNQ3KCNQ2TAS1R3TAS1R1RAB9A
SCHEMBL30622675 0.85 HDAC3 (0.62) TAS1R3TAS1R1RAB9ANPC1USP2
SCHEMBL17141817 0.85 HDAC3 (0.62) TAS1R3TAS1R1RAB9ANPC1USP2
SCHEMBL4898577 0.84 MAPK1 (0.67) KCNQ3KCNQ2RAB9ANPC1USP2
SCHEMBL6582492 0.84 HTT (0.65) KCNQ3KCNQ2TAS1R3TAS1R1RAB9A
SCHEMBL30622701 0.84 HTT (0.65) KCNQ3KCNQ2TAS1R3TAS1R1RAB9A
SCHEMBL6582881 0.83 KCNQ3 (0.54) KCNQ3KCNQ2TAS1R3TAS1R1RAB9A
Hydrochloric Acid SCHEMBL6510141 0.83 HTT (0.63) KCNQ3KCNQ2TAS1R3TAS1R1RAB9A
SCHEMBL2562449 0.82 LMNA (0.67) KCNQ3KCNQ2RAB9ANPC1USP2
SCHEMBL6509070 0.81 POLB (0.65) TAS1R3TAS1R1RAB9ANPC1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed