SCHEMBL6578715

SCHEMBL6578715

COc1ccc(-c2nc(-c3cccc(CN4CCC4)c3)n[nH]2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.62
ADORA1 P30542 2/20 0.62
NR1H2 P55055 1/20 0.55
NR1H3 Q13133 1/20 0.55
DRD2 P14416 2/20 0.54
DRD4 P21917 2/20 0.54
DRD3 P35462 2/20 0.54
CHKA P35790 1/20 0.48
CNR1 P21554 1/20 0.48
CNR2 P34972 1/20 0.48
SIGMAR1 Q99720 2/20 0.46
CHRM3 P20309 1/20 0.46
ACP1 P24666 4/20 0.46
ALDH1A1 P00352 2/20 0.45
POLB P06746 2/20 0.45
LMNA P02545 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
RECQL P46063 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6583869 0.98 ADORA2A (0.65) ADORA2AADORA1NR1H2NR1H3DRD2
Hydrochloric Acid SCHEMBL6578937 0.97 ADORA2A (0.64) ADORA2AADORA1NR1H2NR1H3DRD2
Hydrochloric Acid SCHEMBL6581231 0.96 ADORA2A (0.63) ADORA2AADORA1NR1H2NR1H3DRD2
SCHEMBL6578236 0.94 NR1H2 (0.61) ADORA2AADORA1NR1H2NR1H3DRD2
SCHEMBL6580836 0.89 NR1H2 (0.55) ADORA2AADORA1NR1H2NR1H3DRD2
SCHEMBL6582550 0.89 NR1H2 (0.53) ADORA2AADORA1NR1H2NR1H3DRD2
SCHEMBL6582971 0.89 ADORA2A (0.52) ADORA2AADORA1NR1H2NR1H3DRD2
Hydrochloric Acid SCHEMBL6578786 0.88 ADORA2A (0.61) ADORA2AADORA1NR1H2NR1H3DRD2
Hydrochloric Acid SCHEMBL6580717 0.88 ADORA2A (0.64) ADORA2AADORA1NR1H2NR1H3DRD2
SCHEMBL6580995 0.88 ALDH1A1 (0.52) ADORA2AADORA1NR1H2NR1H3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed