SCHEMBL6582550

SCHEMBL6582550

COc1ccc(-c2nc(-c3cccc(CN4CCN(C=O)CC4)c3)n[nH]2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.53
NR1H3 Q13133 1/20 0.53
ADORA2A P29274 2/20 0.52
ADORA1 P30542 2/20 0.52
DRD4 P21917 3/20 0.50
DRD2 P14416 2/20 0.50
DRD3 P35462 2/20 0.50
LMNA P02545 4/20 0.46
ALDH1A1 P00352 3/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
RECQL P46063 1/20 0.46
KMT2A Q03164 1/20 0.46
CHRM3 P20309 1/20 0.45
SIGMAR1 Q99720 2/20 0.45
BCHE P06276 1/20 0.44
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6578236 0.91 NR1H2 (0.61) NR1H2NR1H3ADORA2AADORA1DRD4
SCHEMBL6578715 0.89 ADORA2A (0.62) NR1H2NR1H3ADORA2AADORA1DRD4
SCHEMBL6583869 0.89 ADORA2A (0.65) NR1H2NR1H3ADORA2AADORA1DRD4
Hydrochloric Acid SCHEMBL6578937 0.88 ADORA2A (0.64) NR1H2NR1H3ADORA2AADORA1DRD4
Hydrochloric Acid SCHEMBL6581231 0.87 ADORA2A (0.63) NR1H2NR1H3ADORA2AADORA1DRD4
SCHEMBL6580995 0.85 ALDH1A1 (0.52) NR1H2NR1H3ADORA2AADORA1DRD4
SCHEMBL6580836 0.85 NR1H2 (0.55) NR1H2NR1H3ADORA2AADORA1DRD4
SCHEMBL6582971 0.84 ADORA2A (0.52) NR1H2NR1H3ADORA2AADORA1DRD4
SCHEMBL6580672 0.83 NR1H2 (0.54) NR1H2NR1H3ADORA2AADORA1DRD4
SCHEMBL6578509 0.82 ADORA2A (0.49) NR1H2NR1H3ADORA2AADORA1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed